SCHEMBL437555

SCHEMBL437555

Nc1c(Cl)cnc2c(Cl)ccc(Cl)c12

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HAVCR2 Q8TDQ0 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.35
NR4A2 P43354 1/20 0.33
DYRK1A Q13627 1/20 0.32
ACHE P22303 1/20 0.32
GAA P10253 1/20 0.31
CYP3A4 P08684 1/20 0.30
TSHR P16473 1/20 0.30
BCL6 P41182 1/20 0.30
DHFR P00374 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL437482 0.84 CYP3A4 (0.35) HAVCR2CYP3A4
SCHEMBL439672 0.82 DYRK1A (0.35) HAVCR2SMN1; SMN2NR4A2DYRK1A
SCHEMBL440283 0.80 DYRK1A (0.39) DYRK1AGAA
SCHEMBL439519 0.80 DYRK1A (0.39) DYRK1AGAA
SCHEMBL440068 0.76 HAVCR2 (0.63) HAVCR2SMN1; SMN2TSHR
SCHEMBL436692 0.74 POLB (0.38) HAVCR2DYRK1ACYP3A4
SCHEMBL439646 0.74 HAVCR2 (0.32) HAVCR2DYRK1A
SCHEMBL441707 0.71 HAVCR2 (0.63) HAVCR2SMN1; SMN2NR4A2DYRK1AACHE
SCHEMBL438820 0.71 HAVCR2 (0.39) HAVCR2SMN1; SMN2NR4A2DYRK1AACHE
SCHEMBL436747 0.69 CYP3A4 (0.32) DYRK1ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed