SCHEMBL437551

SCHEMBL437551

Nc1c(Br)cnc2ccc(Cl)cc12

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 2/20 0.51
ACHE P22303 7/20 0.44
BCHE P06276 4/20 0.44
GRIN1 Q05586 4/20 0.44
GRIN2A Q12879 4/20 0.44
PARP1 P09874 1/20 0.41
MAP4K4 O95819 1/20 0.40
SOS2 Q07890 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
EGFR P00533 1/20 0.39
GABRA1 P14867 1/20 0.38
GABRG2 P18507 1/20 0.38
GABRB3 P28472 1/20 0.38
GABRA5 P31644 1/20 0.38
GABRA3 P34903 1/20 0.38
GABRA2 P47869 1/20 0.38
GABRA6 Q16445 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20424044 0.86 NR4A2 (0.43) NR4A2ACHEBCHEGRIN1GRIN2A
SCHEMBL18658904 0.81 NR4A2 (0.59) NR4A2ACHEBCHEGRIN1GRIN2A
SCHEMBL439464 0.81 NR4A2 (0.55) NR4A2ACHEBCHEGRIN1GRIN2A
SCHEMBL438613 0.81 BCHE (0.45) ACHEBCHEGRIN1GRIN2AGABRA1
SCHEMBL30155016 0.81 NR4A2 (0.59) NR4A2ACHEBCHEGRIN1GRIN2A
SCHEMBL29940962 0.81 NR4A2 (0.46) NR4A2PARP1CYP1A2CYP2D6EGFR
SCHEMBL25668139 0.81 NR4A2 (0.46) NR4A2PARP1CYP1A2CYP2D6EGFR
SCHEMBL439853 0.79 BCHE (0.43) ACHEBCHEGRIN1GRIN2APARP1
SCHEMBL442244 0.79 ACHE (0.43) ACHEBCHEGRIN1GRIN2APARP1
SCHEMBL29392249 0.79 NR4A2 (0.56) NR4A2ACHEBCHEGRIN1GRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed