SCHEMBL442244

SCHEMBL442244

Cc1ccc2ncc(Br)c(N)c2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 5/20 0.43
BCHE P06276 4/20 0.43
GRIN1 Q05586 4/20 0.43
GRIN2A Q12879 4/20 0.43
PARP1 P09874 1/20 0.41
HTR1A P08908 2/20 0.40
ADRA1D P25100 2/20 0.40
ADRA1A P35348 2/20 0.40
ADRA1B P35368 2/20 0.40
HTT P42858 2/20 0.39
POLB P06746 2/20 0.39
LMNA P02545 1/20 0.39
NCOA1 Q15788 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HIF1A Q16665 1/20 0.39
NCOA3 Q9Y6Q9 1/20 0.39
TNF P01375 1/20 0.39
NCK1 P16333 1/20 0.38
BACE1 P56817 1/20 0.38
ELANE P08246 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL437293 0.86 ACHE (0.43) ACHEBCHEGRIN1GRIN2APARP1
SCHEMBL438613 0.81 BCHE (0.45) ACHEBCHEGRIN1GRIN2AHTT
SCHEMBL437551 0.79 NR4A2 (0.51) ACHEBCHEGRIN1GRIN2APARP1
SCHEMBL439853 0.79 BCHE (0.43) ACHEBCHEGRIN1GRIN2APARP1
SCHEMBL440082 0.79 LMNA (0.47) ACHEBCHEGRIN1GRIN2APARP1
SCHEMBL29393479 0.79 PARP1 (0.41) ACHEBCHEGRIN1GRIN2APARP1
SCHEMBL20495272 0.79 PARP1 (0.41) ACHEBCHEGRIN1GRIN2APARP1
SCHEMBL439635 0.78 APP (0.48) ACHEBCHEGRIN1GRIN2AHTR1A
SCHEMBL439366 0.78 ALDH1A1 (0.46) HTTPOLBLMNASMN1; SMN2KDM4E
SCHEMBL437126 0.78 NOS3 (0.38) HTTPOLBSMN1; SMN2BACE1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed