SCHEMBL4375889

SCHEMBL4375889

N=C(N)NCCC[C@H](C(N)=O)N(O)S(=O)(=O)c1ccc(Oc2cccc3ccccc23)nc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 1/20 0.35
MAPK10 P53779 1/20 0.35
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.35
HPGD P15428 1/20 0.35
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
CARM1 Q86X55 1/20 0.34
PRMT6 Q96LA8 1/20 0.34
MCL1 Q07820 1/20 0.33
HTT P42858 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
SIRT2 Q8IXJ6 1/20 0.33
SIRT1 Q96EB6 1/20 0.33
SIRT3 Q9NTG7 1/20 0.33
ADRB2 P07550 1/20 0.33
ADRB1 P08588 1/20 0.33
ADRB3 P13945 1/20 0.33
BMP1 P13497 2/20 0.32
OGG1 O15527 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4372650 0.79 BMP1 (0.51) BMP1ADAMTS4MMP1MMP2MMP14
SCHEMBL4370947 0.79 OPRM1 (0.40)
SCHEMBL1799173 0.76 MMP2 (0.41) HTTBMP1MMP1MMP2MMP13
SCHEMBL4542075 0.75 HPGDS (0.42) SCN9A
SCHEMBL4372258 0.74 F2 (0.41) ALDH1A1BMP1MMP1MMP2MMP13
SCHEMBL1800832 0.73 F2 (0.37) ALDH1A1KDM4EKMT2AMEN1HTT
SCHEMBL1798846 0.71 DAGLA (0.38) ALDH1A1MCL1HTTNPSR1LTA4H
SCHEMBL10528975 0.66 SLC6A4 (0.62) ALDH1A1KDM4EHPGDKMT2A
SCHEMBL4375791 0.65 MMP2 (0.42) HTTLTA4HMMP1MMP2MMP13
SCHEMBL4380644 0.64 MMP2 (0.43) KMT2AMEN1MMP1MMP2MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1461313-B1 HUMAN ADAM-10 INHIBITORS EXELIXIS INC (US) 2009-08-05 EP claimed
EP-1461313-B1 HUMAN ADAM-10 INHIBITORS EXELIXIS INC (US) 2009-08-05 EP disclosed