SCHEMBL4378914

SCHEMBL4378914

O=C(Nc1cccc(Cl)c1)C(=O)c1c(C(F)(F)F)n(Cc2ccc(Cl)cc2Cl)c2ccc(Cl)cc12.O=C(Nc1cccc(Cl)c1)C(=O)c1c(C(F)(F)F)n(Cc2ccc(Cl)cc2Cl)c2ccccc12

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.46
MAPT P10636 6/20 0.43
LMNA P02545 3/20 0.43
ALDH1A1 P00352 1/20 0.43
ALOX12 P18054 1/20 0.43
TP53 P04637 1/20 0.41
NPSR1 Q6W5P4 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
TSHR P16473 1/20 0.41
PMP22 Q01453 1/20 0.41
HIF1A Q16665 1/20 0.41
EPHX2 P34913 1/20 0.40
GAA P10253 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3001227 0.97 THRB (0.47) THRBMAPTLMNAALDH1A1ALOX12
SCHEMBL3006717 0.96 THRB (0.42) THRBMAPTLMNAALDH1A1ALOX12
SCHEMBL3002042 0.92 PLA2G4A (0.43) MAPTLMNAALDH1A1ALOX12NPSR1
SCHEMBL4093752 0.92 LMNA (0.46) THRBMAPTLMNAALDH1A1ALOX12
SCHEMBL4098737 0.91 L3MBTL1 (0.41) THRBMAPTLMNAALDH1A1ALOX12
SCHEMBL4096099 0.90 FAAH (0.46) THRBMAPTLMNAALDH1A1ALOX12
SCHEMBL3001761 0.90 LMNA (0.46) THRBMAPTLMNAALDH1A1ALOX12
SCHEMBL4088421 0.88 PLA2G2A (0.43) THRBMAPTLMNATP53MEN1
SCHEMBL4090425 0.88 CNR1 (0.42) MAPTLMNAALDH1A1ALOX12EPHX2
SCHEMBL3000373 0.87 MAPT (0.43) MAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049520-A2 INDOLE COMPOUNDS Ironwood Pharmaceuticals, Inc. (US) 2009-04-22 EP disclosed
WO-2008019357-A2 INDOLE COMPOUNDS IRONWOOD PHARMACEUTICALS, INC. (US) 2008-02-14 WO disclosed