SCHEMBL437945

SCHEMBL437945

COc1ccc2c(N)c(Br)cnc2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.47
APP P05067 1/20 0.44
GABRA1 P14867 2/20 0.44
GABRG2 P18507 2/20 0.44
GABRB3 P28472 2/20 0.44
GABRA5 P31644 2/20 0.44
GABRA3 P34903 2/20 0.44
GABRA6 Q16445 2/20 0.44
HTR1A P08908 2/20 0.43
ADRA1D P25100 2/20 0.43
ADRA1A P35348 2/20 0.43
ADRA1B P35368 2/20 0.43
FERMT2 Q96AC1 1/20 0.43
HPGDS O60760 2/20 0.42
EGFR P00533 3/20 0.42
GABRA2 P47869 1/20 0.42
PDGFRB P09619 1/20 0.40
PDGFRA P16234 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP3A4 P08684 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL439635 0.87 APP (0.48) ACHEAPPGABRA1GABRG2GABRB3
SCHEMBL440277 0.81 ACHE (0.50) ACHEAPPGABRA1GABRG2GABRB3
SCHEMBL20495237 0.81 GABRA1 (0.44) ACHEGABRA1GABRG2GABRB3GABRA5
SCHEMBL29392911 0.81 GABRA1 (0.44) ACHEGABRA1GABRG2GABRB3GABRA5
SCHEMBL23896032 0.81 GABRA1 (0.44) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL439912 0.80 ALOX5AP (0.42) HPGDSALDH1A1CYP3A4NPC1RAB9A
SCHEMBL437293 0.78 ACHE (0.43) ACHEHTR1AADRA1DADRA1AADRA1B
SCHEMBL437952 0.78 ACHE (0.45) ACHEKMT2A
SCHEMBL21358444 0.77 PDPK1 (0.47) ACHEEGFR
SCHEMBL30368021 0.75 PIM1 (0.45) ACHEAPPGABRA1GABRG2GABRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed