SCHEMBL437293

SCHEMBL437293

Cc1ccc2c(N)c(Br)cnc2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 4/20 0.43
BCHE P06276 4/20 0.42
GRIN1 Q05586 3/20 0.42
GRIN2A Q12879 3/20 0.42
CHEK1 O14757 1/20 0.41
PARP1 P09874 1/20 0.41
PIM1 P11309 1/20 0.41
RPS6KA3 P51812 1/20 0.41
HTR1A P08908 2/20 0.39
ADRA1D P25100 2/20 0.39
ADRA1A P35348 2/20 0.39
ADRA1B P35368 2/20 0.39
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
GAA P10253 1/20 0.38
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38
TP53 P04637 1/20 0.38
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL442244 0.86 ACHE (0.43) ACHEBCHEGRIN1GRIN2APARP1
SCHEMBL437952 0.81 ACHE (0.45) ACHE
SCHEMBL12210442 0.81 ACHE (0.49) ACHEBCHEGRIN1GRIN2ACHEK1
SCHEMBL25544293 0.79 CHEK1 (0.41) CHEK1PARP1PIM1RPS6KA3HTR1A
SCHEMBL442268 0.79 ACHE (0.46) ACHEBCHEGRIN1GRIN2ACHEK1
SCHEMBL439004 0.79 ACHE (0.43) ACHE
SCHEMBL437945 0.78 ACHE (0.47) ACHEHTR1AADRA1DADRA1AADRA1B
SCHEMBL437126 0.78 NOS3 (0.38) KDM4EALDH1A1GAATP53CYP3A4
SCHEMBL437195 0.76 UHRF1 (0.35) PSMB5NOS3NOS2
SCHEMBL437067 0.75 MAOB (0.46) PARP1NOS3NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed