SCHEMBL4380448

SCHEMBL4380448

CN1C(N)=Nc2nc(-c3c(OCCN4CCCC4)cccc3C(F)(F)F)ccc2C1N

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.43
PTGS2 P35354 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C19 P33261 1/20 0.43
HSD17B10 Q99714 1/20 0.43
NOS3 P29474 3/20 0.39
NOS1 P29475 3/20 0.39
NOS2 P35228 3/20 0.39
ALDH1A1 P00352 2/20 0.39
DRD2 P14416 4/20 0.38
TDP1 Q9NUW8 1/20 0.38
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
HTR2B P41595 1/20 0.37
POLB P06746 1/20 0.37
AXL P30530 1/20 0.37
BACE1 P56817 1/20 0.37
MCHR1 Q99705 1/20 0.36
HTR1A P08908 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4373757 0.92 HTR2A (0.38) DRD2HTR2AHTR2CHTR2B
SCHEMBL4384328 0.90 PTPN1 (0.36) LTA4HPTGS2DRD2HTR2AHTR2C
SCHEMBL4381198 0.89 PTPN1 (0.38) LTA4HPTGS2ALDH1A1DRD2HTR2A
SCHEMBL4384579 0.88 PTPN1 (0.37) HTR2AHTR2CHTR2B
SCHEMBL4381287 0.87 CTSS (0.36) NOS3NOS1NOS2ALDH1A1DRD2
SCHEMBL4378503 0.85 PTPN1 (0.48) HTR2AHTR2CHTR2B
SCHEMBL3742273 0.83 PTPN1 (0.36) HTR2AHTR2CHTR2B
SCHEMBL4373580 0.83 MCHR1 (0.36) MCHR1
SCHEMBL4379622 0.82 PTPN1 (0.37) HTR2AHTR2CHTR2BMCHR1HTR1A
SCHEMBL3732060 0.81 PTPN1 (0.52) HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910359-B1 PYRIDO [2 , 3-D]PYRIMIDINE-2 , 4-DIAMINE COMPOUNDS AS PTPlB INHIBITORS HOFFMANN LA ROCHE (CH) 2009-11-18 EP claimed