SCHEMBL4384328

SCHEMBL4384328

CCCOc1cccc(C(F)(F)F)c1-c1ccc2c(n1)N=C(N)N(C)C2N

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 2/20 0.36
MCHR1 Q99705 1/20 0.34
HTR2A P28223 3/20 0.32
HTR2C P28335 3/20 0.32
HTR2B P41595 2/20 0.32
DRD2 P14416 5/20 0.32
IKBKB O14920 1/20 0.32
HSP90AA1 P07900 1/20 0.31
HSP90AB1 P08238 1/20 0.31
TLR8 Q9NR97 1/20 0.31
CTSS P25774 1/20 0.31
CTSK P43235 1/20 0.31
KCNH2 Q12809 1/20 0.30
LTA4H P09960 1/20 0.30
PTGS2 P35354 1/20 0.30
PDE3B Q13370 1/20 0.30
PDE3A Q14432 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4384579 0.92 PTPN1 (0.37) PTPN1HTR2AHTR2CHTR2BIKBKB
SCHEMBL4381198 0.91 PTPN1 (0.38) PTPN1HTR2AHTR2CHTR2BDRD2
SCHEMBL4380448 0.90 LTA4H (0.43) MCHR1HTR2AHTR2CHTR2BDRD2
SCHEMBL4381287 0.90 CTSS (0.36) PTPN1DRD2CTSSCTSK
SCHEMBL4373757 0.87 HTR2A (0.38) PTPN1HTR2AHTR2CHTR2BDRD2
SCHEMBL4378502 0.87 MCHR1 (0.36) MCHR1IKBKBTLR8
SCHEMBL4378503 0.87 PTPN1 (0.48) PTPN1HTR2AHTR2CHTR2BHSP90AA1
SCHEMBL3742273 0.85 PTPN1 (0.36) PTPN1HTR2AHTR2CHTR2BTLR8
SCHEMBL4379622 0.84 PTPN1 (0.37) PTPN1MCHR1HTR2AHTR2CHTR2B
SCHEMBL4389955 0.83 PTPN1 (0.51) PTPN1HTR2AHTR2CHTR2BDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910359-B1 PYRIDO [2 , 3-D]PYRIMIDINE-2 , 4-DIAMINE COMPOUNDS AS PTPlB INHIBITORS HOFFMANN LA ROCHE (CH) 2009-11-18 EP claimed