SCHEMBL4381198

SCHEMBL4381198

COCCOc1cccc(C(F)(F)F)c1-c1ccc2c(n1)N=C(N)N(C)C2N

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 2/20 0.38
AR P10275 2/20 0.36
HTR2A P28223 2/20 0.33
HTR2C P28335 2/20 0.33
HTR2B P41595 1/20 0.33
MIF P14174 1/20 0.32
DRD2 P14416 4/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GLA P06280 1/20 0.32
GAA P10253 1/20 0.32
HPGD P15428 1/20 0.32
HSP90AA1 P07900 1/20 0.31
HSP90AB1 P08238 1/20 0.31
ADORA2A P29274 1/20 0.30
KCNH2 Q12809 1/20 0.30
LTA4H P09960 1/20 0.30
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4384328 0.91 PTPN1 (0.36) PTPN1HTR2AHTR2CHTR2BDRD2
SCHEMBL4384579 0.89 PTPN1 (0.37) PTPN1HTR2AHTR2CHTR2B
SCHEMBL4380448 0.89 LTA4H (0.43) HTR2AHTR2CHTR2BDRD2ALDH1A1
SCHEMBL4381287 0.89 CTSS (0.36) PTPN1DRD2KDM4EALDH1A1
SCHEMBL4378503 0.88 PTPN1 (0.48) PTPN1ARHTR2AHTR2CHTR2B
SCHEMBL4373757 0.87 HTR2A (0.38) PTPN1HTR2AHTR2CHTR2BDRD2
SCHEMBL3742273 0.85 PTPN1 (0.36) PTPN1HTR2AHTR2CHTR2B
SCHEMBL4379622 0.83 PTPN1 (0.37) PTPN1HTR2AHTR2CHTR2B
SCHEMBL4524489 0.83 AR (0.40) ARHTR2AHTR2CHTR2BDRD2
SCHEMBL4389955 0.83 PTPN1 (0.51) PTPN1HTR2AHTR2CHTR2BDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910359-B1 PYRIDO [2 , 3-D]PYRIMIDINE-2 , 4-DIAMINE COMPOUNDS AS PTPlB INHIBITORS HOFFMANN LA ROCHE (CH) 2009-11-18 EP claimed