SCHEMBL4383375

SCHEMBL4383375

Nc1c(Cl)cc(Cl)cc1C1=NCCN1

nearest known ligand 0.61

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 9/20 0.50
LMNA P02545 1/20 0.45
RECQL P46063 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10471223 0.80 CYP3A4 (0.41) NISCHLMNARECQL
SCHEMBL11155987 0.80 NISCH (0.50) NISCHLMNARECQL
SCHEMBL11301090 0.77 LMNA (0.53) NISCHLMNARECQL
SCHEMBL11285481 0.73 NISCH (0.54) NISCHLMNARECQL
SCHEMBL30982286 0.71 LMNA (0.54) NISCHLMNARECQL
SCHEMBL10818104 0.71 ALDH1A1 (0.48) RECQL
SCHEMBL11517317 0.70 NISCH (0.67) NISCHLMNARECQL
SCHEMBL18824619 0.70 LMNA (0.53) NISCHLMNARECQL
SCHEMBL8239326 0.70 NISCH (0.57) NISCHLMNARECQL
SCHEMBL2949149 0.68 NISCH (0.62) NISCH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7629463-B2 Ortho-heterocyclic substituted aryl amides for controlling invertebrate pests E. I. DU PONT DE NEMOURS AND COMPANY (US) 2009-12-08 US disclosed
EP-1435785-B1 IMINOBENZOXAZINES, IMINOBENZOTHIAZINES AND IMINOQUINAZOLINES FOR CONTROLLING INVERTEBRATE PESTS DU PONT (US) 2008-12-31 EP disclosed
US-20080132524-A1 Ortho-heterocyclic substituted aryl amides for controlling invertebrate pests CLARK DAVID ALAN 2008-06-05 US disclosed
US-7375232-B2 Ortho-heterocyclic substituted aryl amides for controlling invertebrate pests E.I. DU PONT DE NEMOURS AND COMPANY (US) 2008-05-20 US disclosed
US-7326704-B2 Iminobenzoxazines, iminobenzthiazines and iminoquinazolines for controlling invertebrate pests E.I. DUPONT DE NEMOURS AND COMPANY (US) 2008-02-05 US disclosed
US-7148217-B2 Iminobenzoxazines, iminobenzthiazines and iminoquinazolines for controlling invertebrate pests E. I. DU PONT DE NEMOURS AND COMPANY (US) 2006-12-12 US disclosed
US-20060258649-A1 Iminobenzoxazines, iminobenzthiazines and iminoquinazolines for controlling invertebrate pests SELBY THOMAS P 2006-11-16 US disclosed
EP-1417204-B1 ORTHO-HETEROCYCLIC SUBSTITUTED ARYL AMIDES FOR CONTROLLING INVERTEBRATE PESTS DU PONT (US) 2006-01-18 EP disclosed
US-20040242645-A1 Ortho-heterocyclic substituted aryl amides for controlling invertebrate pests E. I. DU PONT DE NEMOURS AND COMPANY 2004-12-02 US disclosed
US-20040214828-A1 Iminobenzoxazines, iminobenzthiazines and iminoquinazolines for controlling invertebrate pests E.I. DU PONT DE NEMOURS AND COMPANY 2004-10-28 US disclosed
EP-1417204-A1 ORTHO-HETEROCYCLIC SUBSTITUTED ARYL AMIDES FOR CONTROLLING INVERTEBRATE PESTS E. I. du Pont de Nemours and Company (US) 2004-05-12 EP disclosed
WO-2003016304-A1 ORTHO-HETEROCYCLIC SUBSTITUTED ARYL AMIDES FOR CONTROLLING INVERTEBRATE PESTS E. I. DU PONT DE NEMOURS AND COMPANY (US) 2003-02-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080132524-A1 Ortho-heterocyclic substituted aryl amides for controlling invertebrate pests AOC2, DDT, CBR3 NISCH 53/4885LMNA 4791/4885RECQL 504/4885
US-20040214828-A1 Iminobenzoxazines, iminobenzthiazines and iminoquinazolines for controlling invertebrate pests NR0B1, IPO5, RER1 NISCH 19/4885LMNA 1088/4885RECQL 98/4885
US-20040242645-A1 Ortho-heterocyclic substituted aryl amides for controlling invertebrate pests AOC2, OLA1, AOC3 NISCH 17/4885LMNA 3892/4885RECQL 821/4885
US-20060258649-A1 Iminobenzoxazines, iminobenzthiazines and iminoquinazolines for controlling invertebrate pests NR0B1, NR1I2, NR0B2 NISCH 166/4885LMNA 1633/4885RECQL 160/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.