SCHEMBL4385912

SCHEMBL4385912

Cc1c(O)ccnc1C#N

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLCG1 P19174 1/20 0.35
AR P10275 1/20 0.34
KDM4E B2RXH2 1/20 0.32
MAPK1 P28482 1/20 0.32
TRPA1 O75762 1/20 0.32
ATM Q13315 1/20 0.32
CDK4 P11802 2/20 0.31
CDK2 P24941 2/20 0.31
ERBB2 P04626 1/20 0.31
MAPT P10636 1/20 0.31
ELANE P08246 1/20 0.31
KDM4C Q9H3R0 1/20 0.30
NOS3 P29474 1/20 0.30
NOS2 P35228 1/20 0.30
CHEK1 O14757 1/20 0.30
ABL1 P00519 1/20 0.30
PDGFRB P09619 1/20 0.30
PDGFRA P16234 1/20 0.30
FLT1 P17948 1/20 0.30
GRK5 P34947 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6170131 0.78 NOS3 (0.46) PLCG1KDM4EMAPK1ERBB2MAPT
SCHEMBL7788094 0.78 PLCG1 (0.33) PLCG1KDM4EMAPK1CDK2MAPT
SCHEMBL17570530 0.77 TSHR (0.37) PLCG1ARCDK2ERBB2MAPT
SCHEMBL4385911 0.75 ALDH1A1 (0.36) PLCG1TRPA1ERBB2MAPTELANE
SCHEMBL25299754 0.75 NTRK1 (0.33) PLCG1ERBB2MAPTNOS3NOS2
SCHEMBL19798237 0.75 GSK3A (0.33) PLCG1KDM4CGSK3AGSK3B
SCHEMBL2671146 0.75 ALDH1A1 (0.40) PLCG1KDM4EMAPK1ERBB2MAPT
SCHEMBL19774234 0.75 NOS3 (0.35) PLCG1KDM4ENOS3NOS2
SCHEMBL28371872 0.73 KDM4E (0.41) PLCG1KDM4EMAPTKDM4C
SCHEMBL6649929 0.72 ROCK2 (0.45) KDM4EMAPK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009119880-A1 SUBSTITUTED PYRAZOLE DERIVATIVES AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-10-01 WO disclosed