SCHEMBL4387186

SCHEMBL4387186

Cc1ccc(Oc2ncccc2C(=O)NC2CCCCn3c2nc(-c2ccncc2)cc3=O)cc1

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.56
GAA P10253 1/20 0.43
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
KDM4E B2RXH2 1/20 0.38
UGCG Q16739 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4388471 0.92 KDM4E (0.47) L3MBTL1GAAKDM4EUGCG
SCHEMBL4953302 0.89 L3MBTL1 (0.53) L3MBTL1GAAMEN1KMT2AKDM4E
SCHEMBL4952879 0.88 MEN1 (0.47) L3MBTL1MEN1KMT2AKDM4E
SCHEMBL4383616 0.86 MEN1 (0.47) L3MBTL1GAAMEN1KMT2A
SCHEMBL4391863 0.83 MAPT (0.40) GAAMEN1KMT2A
SCHEMBL4391283 0.83 CYP2C9 (0.39) L3MBTL1GAAMEN1KMT2AKDM4E
SCHEMBL4385766 0.83 RAB9A (0.51) L3MBTL1MEN1KMT2AKDM4E
SCHEMBL2065962 0.82 KMT2A (0.46) MEN1KMT2AKDM4E
SCHEMBL4377844 0.82 MEN1 (0.45) L3MBTL1GAAMEN1KMT2A
SCHEMBL4393751 0.81 KDM4E (0.46) L3MBTL1KDM4EUGCG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121635-A2 SUBSTITUTED HETEROARYL PYRIDOPYRIMIDONE DERIVATIVES Sanofi-Aventis (FR) 2009-11-25 EP claimed
WO-2008078196-A2 SUBSTITUTED HETEROARYL PYRIDOPYRIMIDONE DERIVATIVES SANOFI-AVENTIS (FR) 2008-07-03 WO claimed
EP-1939187-A1 Substituted heteroaryl pyridopyrimidone derivatives Sanofi-Aventis (FR) 2008-07-02 EP claimed
US-8198287-B2 Substituted heteroaryl pyridopyrimidone derivatives SANOFI-AVENTIS (FR) 2012-06-12 US disclosed
EP-2121635-A2 SUBSTITUTED HETEROARYL PYRIDOPYRIMIDONE DERIVATIVES Sanofi-Aventis (FR) 2009-11-25 EP disclosed
WO-2008078196-A2 SUBSTITUTED HETEROARYL PYRIDOPYRIMIDONE DERIVATIVES SANOFI-AVENTIS (FR) 2008-07-03 WO disclosed
EP-1939187-A1 Substituted heteroaryl pyridopyrimidone derivatives Sanofi-Aventis (FR) 2008-07-02 EP disclosed