SCHEMBL438818

SCHEMBL438818

Nc1c(C(=O)O)cnc2cc(C(F)(F)F)ccc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.53
HPGD P15428 3/20 0.53
KDM4E B2RXH2 2/20 0.53
HSD17B10 Q99714 2/20 0.53
CSF1R P07333 1/20 0.46
ALOX5AP P20292 1/20 0.46
FEN1 P39748 1/20 0.46
PARP1 P09874 1/20 0.44
MEN1 O00255 1/20 0.44
CYP1A2 P05177 1/20 0.44
ALOX12 P18054 1/20 0.44
KMT2A Q03164 1/20 0.44
HAVCR2 Q8TDQ0 1/20 0.43
SORT1 Q99523 4/20 0.42
TBK1 Q9UHD2 1/20 0.42
THRB P10828 1/20 0.41
MAP4K4 O95819 2/20 0.41
PLK4 O00444 1/20 0.41
DYRK3 O43781 1/20 0.41
PRKD3 O94806 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL439948 0.89 ALDH1A1 (0.53) ALDH1A1HPGDKDM4EHSD17B10CSF1R
SCHEMBL1644467 0.86 THRB (0.46) ALDH1A1HPGDKDM4EHSD17B10CSF1R
SCHEMBL30592902 0.84 ALDH1A1 (0.46) ALDH1A1HPGDKDM4EHSD17B10CSF1R
SCHEMBL3887756 0.84 ALDH1A1 (0.46) ALDH1A1HPGDKDM4EHSD17B10CSF1R
Hydrochloric Acid SCHEMBL11870232 0.83 ALDH1A1 (0.45) ALDH1A1HPGDKDM4EHSD17B10CSF1R
SCHEMBL4466003 0.83 SORT1 (0.46) ALDH1A1HPGDKDM4EHSD17B10CSF1R
SCHEMBL437005 0.81 THRB (0.60) ALDH1A1KDM4EKMT2ATHRB
SCHEMBL438745 0.81 KEAP1 (0.49) ALDH1A1KDM4ECSF1RMEN1KMT2A
SCHEMBL27855175 0.79 CSF1R (0.51) CSF1RPARP1KMT2ATHRBMAP4K4
SCHEMBL5757387 0.78 KDM4C (0.51) ALDH1A1HPGDKDM4EHSD17B10PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed