SCHEMBL438849

SCHEMBL438849

CCCc1cc(N)c2cc(F)cc(F)c2n1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.41
NOS1 P29475 1/20 0.41
NOS2 P35228 1/20 0.41
MCHR1 Q99705 13/20 0.40
BACE1 P56817 1/20 0.38
EIF4A1 P60842 1/20 0.35
NPC1 O15118 1/20 0.35
TP53 P04637 1/20 0.35
PKM P14618 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HSD17B10 Q99714 1/20 0.35
SREBF2 Q12772 1/20 0.35
PDE10A Q9Y233 1/20 0.34
ASIC3 Q9UHC3 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL436520 0.81 CYP2D6 (0.41) NOS3NOS1NOS2MCHR1BACE1
SCHEMBL436015 0.78 NOS3 (0.39) NOS3NOS1NOS2MCHR1BACE1
SCHEMBL437488 0.76 MCHR1 (0.58) MCHR1ASIC3
SCHEMBL436969 0.74 NR4A2 (0.46) NOS3NOS1NOS2PKMRAB9A
SCHEMBL439708 0.73 MCHR1 (0.43) NOS3NOS1NOS2MCHR1BACE1
SCHEMBL439432 0.73 MCHR1 (0.49) NOS3NOS1NOS2MCHR1ASIC3
SCHEMBL437498 0.72 NOS2 (0.50) NOS3NOS1NOS2MCHR1BACE1
SCHEMBL438834 0.72 NOS2 (0.50) NOS3NOS1NOS2MCHR1BACE1
SCHEMBL440057 0.72 NOS2 (0.42) NOS3NOS1NOS2MCHR1BACE1
SCHEMBL438887 0.72 MCHR1 (0.44) NOS3NOS1NOS2MCHR1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed