SCHEMBL440057

SCHEMBL440057

CCCc1cc(N)c2cc(Br)cc(C)c2n1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 2/20 0.42
NOS3 P29474 1/20 0.42
NOS1 P29475 1/20 0.42
MCHR1 Q99705 13/20 0.41
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
BACE1 P56817 1/20 0.36
ASIC3 Q9UHC3 1/20 0.34
NQO2 P16083 1/20 0.34
PARP1 P09874 1/20 0.34
PARP2 Q9UGN5 1/20 0.34
PARP4 Q9UKK3 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL438887 0.82 MCHR1 (0.44) NOS2NOS3NOS1MCHR1KDM4E
SCHEMBL437498 0.79 NOS2 (0.50) NOS2NOS3NOS1MCHR1KDM4E
SCHEMBL442077 0.77 NR4A2 (0.45) KDM4EALDH1A1NQO2PARP1PARP2
SCHEMBL440305 0.77 MCHR1 (0.58) MCHR1ASIC3
SCHEMBL437578 0.76 MCHR1 (0.43) NOS2NOS3NOS1MCHR1ASIC3
SCHEMBL438834 0.76 NOS2 (0.50) NOS2NOS3NOS1MCHR1KDM4E
SCHEMBL440069 0.75 NOS2 (0.41) NOS2NOS3NOS1MCHR1ALDH1A1
SCHEMBL437548 0.74 MCHR1 (0.49) NOS2NOS3NOS1MCHR1KDM4E
SCHEMBL440380 0.73 ALDH1A1 (0.49) NOS2NOS3NOS1MCHR1KDM4E
SCHEMBL438849 0.72 NOS3 (0.41) NOS2NOS3NOS1MCHR1BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed