SCHEMBL4392546

SCHEMBL4392546

O=Cc1cccc(-c2cc3sc(Cl)cc3c(N3CCOCC3)n2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKDC P78527 2/20 0.43
ALDH3A1 P30838 1/20 0.41
ALDH1A3 P47895 1/20 0.41
ALDH1A1 P00352 4/20 0.41
MAPK1 P28482 3/20 0.41
KDM4E B2RXH2 2/20 0.41
HPGD P15428 2/20 0.41
HSD17B10 Q99714 2/20 0.41
LMNA P02545 1/20 0.41
TSHR P16473 1/20 0.41
PIM2 Q9P1W9 1/20 0.39
PIK3CA P42336 8/20 0.39
MTOR P42345 3/20 0.39
PIK3R1 P27986 4/20 0.38
PIK3C2A O00443 1/20 0.38
PIK3C2B O00750 1/20 0.38
PIK3C3 Q8NEB9 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
USP2 O75604 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4554179 0.84 KMO (0.47) PRKDCALDH1A1MAPK1KDM4EHPGD
SCHEMBL4554583 0.84 PIK3CA (0.47) PRKDCALDH1A1MAPK1KDM4EHPGD
SCHEMBL4555862 0.80 BRAF (0.51) PRKDCALDH1A1KDM4EPIK3CAMTOR
SCHEMBL4252078 0.78 NPC1 (0.46) PIK3CAMTORPIK3R1PIK3C2BMEN1
SCHEMBL1864535 0.78 SMN1; SMN2 (0.38) ALDH3A1ALDH1A3ALDH1A1MAPK1KDM4E
SCHEMBL4566064 0.76 PIK3CA (0.39) PRKDCALDH1A1MAPK1KDM4EHPGD
SCHEMBL3993337 0.75 PIK3CA (0.51) PRKDCALDH3A1ALDH1A3MAPK1HSD17B10
SCHEMBL1860764 0.72 NCF1 (0.45) PRKDCALDH1A1MAPK1KDM4EHPGD
SCHEMBL4565478 0.72 KDM4E (0.38) ALDH1A1MAPK1KDM4EHPGDHSD17B10
SCHEMBL1865304 0.71 PIKFYVE (0.51) PRKDCALDH3A1ALDH1A3ALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2046799-A1 PHOSPHOINOSITIDE 3-KINASE INHIBITOR COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Genentech, Inc. (US) 2009-04-15 EP disclosed
WO-2007127183-A1 PHOSPHOINOSITIDE 3-KINASE INHIBITOR COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GENENTECH, INC. (US) 2007-11-08 WO disclosed