SCHEMBL4393666

SCHEMBL4393666

Cn1[c]nnc1-c1cnccn1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 6/20 0.40
P2RX7 Q99572 1/20 0.40
ALDH1A1 P00352 6/20 0.39
NPC1 O15118 4/20 0.39
TDP1 Q9NUW8 2/20 0.39
USP2 O75604 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
KDM4E B2RXH2 1/20 0.39
CYP1A2 P05177 1/20 0.37
TSHR P16473 2/20 0.36
MAPT P10636 1/20 0.36
PKM P14618 1/20 0.36
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HSD17B10 Q99714 1/20 0.36
GFER P55789 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8629186 0.75 NPC1 (0.50) RAB9AALDH1A1NPC1TDP1L3MBTL1
SCHEMBL18912013 0.70 RAB9A (0.51) RAB9AP2RX7ALDH1A1NPC1TDP1
SCHEMBL8629217 0.70 ALDH1A1 (0.47) RAB9AALDH1A1NPC1USP2L3MBTL1
SCHEMBL4398572 0.69 P2RX7 (0.41) RAB9AP2RX7ALDH1A1NPC1TDP1
SCHEMBL11126232 0.68 CYP1A2 (0.40) RAB9AP2RX7ALDH1A1NPC1TDP1
SCHEMBL4701736 0.68 RAB9A (0.49) RAB9AP2RX7ALDH1A1NPC1TDP1
SCHEMBL9007472 0.67 CYP1A2 (0.39) RAB9AP2RX7ALDH1A1NPC1TDP1
SCHEMBL29598957 0.66 NISCH (0.50) RAB9AP2RX7ALDH1A1NPC1KDM4E
SCHEMBL29454745 0.66 NISCH (0.50) RAB9AP2RX7ALDH1A1NPC1KDM4E
SCHEMBL78566 0.66 NISCH (0.50) RAB9AP2RX7ALDH1A1NPC1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1778684-B1 4-PIPERAZINYL-PYRIMIDINE COMPOUNDS SUITABLE FOR TREATING DISORDERS THAT RESPOND TO MODULATION OF THE DOPAMINE D<sb>3</sb> RECEPTOR ABBOTT GMBH & CO KG (DE) 2009-12-16 EP disclosed