SCHEMBL4394775

SCHEMBL4394775

CC(C)NC(=O)c1cnccc1C(F)(F)F

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.56
POLB P06746 1/20 0.56
ALDH1A1 P00352 1/20 0.47
MAPT P10636 1/20 0.45
NTRK1 P04629 1/20 0.44
DGAT2 Q96PD7 1/20 0.43
MLYCD O95822 1/20 0.43
NPSR1 Q6W5P4 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
KLRK1 P26718 5/20 0.41
MICA Q29983 5/20 0.41
RAET1L Q5VY80 5/20 0.41
GABRA5 P31644 1/20 0.41
KDM5A P29375 1/20 0.41
GAA P10253 1/20 0.41
CHRM2 P08172 1/20 0.41
GRM5 P41594 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
RBP4 P02753 1/20 0.41
CTSS P25774 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21571478 0.85 NPC1 (0.60) NPC1POLBALDH1A1MAPTNTRK1
SCHEMBL22048232 0.85 NPC1 (0.50) NPC1POLBALDH1A1MAPTNTRK1
SCHEMBL18705673 0.85 NPC1 (0.50) NPC1POLBALDH1A1MAPTNTRK1
SCHEMBL18705566 0.84 NPC1 (0.49) NPC1POLBALDH1A1MAPTNTRK1
SCHEMBL3759581 0.83 POLB (0.59) NPC1POLBALDH1A1MAPTNTRK1
SCHEMBL29100737 0.82 NPC1 (0.53) NPC1POLBALDH1A1MAPTNTRK1
SCHEMBL30620180 0.82 NPC1 (0.53) NPC1POLBALDH1A1MAPTNTRK1
SCHEMBL5106559 0.82 NPC1 (0.53) NPC1POLBALDH1A1MAPTNTRK1
SCHEMBL15244373 0.82 NPC1 (0.62) NPC1POLBALDH1A1MAPTNTRK1
SCHEMBL3770167 0.82 ALDH1A1 (0.51) NPC1POLBALDH1A1MAPTNTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7629348-B2 Heterocyclic amide and imine derivatives, processes for their preparation, compositions comprising them and their use as pesticides MERIAL LIMITED (US) 2009-12-08 US disclosed
US-20080139627-A1 Heterocyclic amide and imine derivatives, processes for their preparation, compositions comprising them and their use as pesticides BECKMANN MARION 2008-06-12 US disclosed
US-20080097099-A1 Heterocyclic amide and imine derivatives, processes for their preparation, compositions comprising them and their use as pesticides BECKMANN MARION 2008-04-24 US disclosed
EP-1432313-B1 N-THIO-NICOTINAMIDE DERIVATIVES AND RELATED COMPOUNDS FOR USE AS PESTICIDES MERIAL LTD (US) 2008-01-23 EP disclosed
US-7235571-B2 Heterocyclic amide and imine derivatives, processes for their preparation, compositions comprising them and their use as pesticides MERIAL LIMITED (US) 2007-06-26 US disclosed
US-20040192712-A1 Heterocyclic amide and imine derivatives, processes for their preparation, compositions comprising them and their use as pesticides MERIAL LIMITED 2004-09-30 US disclosed
US-20030119852-A1 Heterocyclic amide and imine derivatives, processes for their preparation, compositions, comprising them and their use as pesticides BAYER CROPSCIENCE GMBH (GE) 2003-06-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080139627-A1 Heterocyclic amide and imine derivatives, processes for their preparation, compositions comprising them and their use as pesticides ACHE, DDT, PIR NPC1 4481/4885POLB 4499/4885ALDH1A1 1482/4885
US-20040192712-A1 Heterocyclic amide and imine derivatives, processes for their preparation, compositions comprising them and their use as pesticides ACHE, DDT, PIR NPC1 3901/4885POLB 4539/4885ALDH1A1 517/4885
US-20030119852-A1 Heterocyclic amide and imine derivatives, processes for their preparation, compositions, comprising them and their use as pesticides ACHE, DDT, PIR NPC1 4068/4885POLB 4414/4885ALDH1A1 504/4885
US-20080097099-A1 Heterocyclic amide and imine derivatives, processes for their preparation, compositions comprising them and their use as pesticides ACHE, DDT, PIR NPC1 4551/4885POLB 4317/4885ALDH1A1 1101/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.