SCHEMBL4399337

SCHEMBL4399337

COc1ccc2c(COc3cccc4[nH]c(OC(=O)NC5CCN(C[C@H](C)N6CCC(O)CC6)CC5)cc34)coc2c1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.41
MCHR1 Q99705 5/20 0.38
KCNH2 Q12809 3/20 0.36
ALDH1A1 P00352 2/20 0.36
LTA4H P09960 3/20 0.35
SLC2A1 P11166 1/20 0.35
HTR1A P08908 2/20 0.35
ACHE P22303 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
MAPT P10636 1/20 0.34
ADRB2 P07550 1/20 0.34
ADRB1 P08588 1/20 0.34
ADRB3 P13945 1/20 0.34
SLC6A4 P31645 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4404545 0.92 MAOB (0.39) MAOBMCHR1KCNH2ALDH1A1LTA4H
SCHEMBL4400742 0.92 MCHR1 (0.36) MAOBMCHR1KCNH2SLC2A1HTR1A
Hydrochloric Acid SCHEMBL4403801 0.92 HTR1A (0.37) MCHR1KCNH2HTR1A
SCHEMBL4401792 0.92 DRD2 (0.35) MAOBHTR1AACHESLC6A4
SCHEMBL4401840 0.92 MAOB (0.44) MAOBMCHR1ALDH1A1LTA4HHTR1A
Hydrochloric Acid SCHEMBL4396448 0.91 SOS1 (0.33) MAOBMCHR1KCNH2LTA4HHTR1A
Hydrochloric Acid SCHEMBL4396591 0.90 HTR1A (0.34) MCHR1ALDH1A1HTR1ASLC6A4
SCHEMBL914491 0.90 MAOB (0.43) MAOBMCHR1KCNH2ALDH1A1LTA4H
Hydrochloric Acid SCHEMBL4405664 0.89 HTR1A (0.35) MCHR1SLC2A1HTR1AADRB2ADRB1
Hydrochloric Acid SCHEMBL4396450 0.88 SOS1 (0.36) MAOBMCHR1KCNH2HTR1ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720859-B1 CHEMOKINE RECEPTOR ANTAGONISTS NOVARTIS AG (CH) 2009-12-23 EP claimed