SCHEMBL4399700

SCHEMBL4399700

CCOC(=O)C1C(=O)c2cc(C=CC(N)=O)ccc2N(CC)C1=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
TTR P02766 1/20 0.36
DPP4 P27487 1/20 0.36
NPC1 O15118 5/20 0.35
RAB9A P51151 5/20 0.35
POLB P06746 1/20 0.35
IDO1 P14902 1/20 0.34
TDO2 P48775 1/20 0.34
SMN1; SMN2 Q16637 4/20 0.34
LMNA P02545 2/20 0.34
MAPT P10636 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
HTT P42858 1/20 0.34
KMT2A Q03164 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
MAOB P27338 1/20 0.34
GAA P10253 1/20 0.34
RXRA P19793 3/20 0.33
CA12 O43570 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4399697 1.00 ALDH1A1 (0.38) ALDH1A1TTRDPP4NPC1RAB9A
SCHEMBL4386782 0.79 ALDH1A1 (0.40) ALDH1A1MAPTKDM4EMEN1KMT2A
SCHEMBL4385104 0.68 BRD4 (0.38) ALDH1A1IDO1MEN1KMT2AGAA
SCHEMBL30099632 0.66 GABRG2 (0.41) ALDH1A1IDO1TDO2SMN1; SMN2MAPT
SCHEMBL23609872 0.66 GABRG2 (0.41) ALDH1A1IDO1TDO2SMN1; SMN2MAPT
SCHEMBL2743830 0.66 ALDH1A1 (0.47) ALDH1A1SMN1; SMN2MAPTKDM4EMEN1
SCHEMBL5059322 0.65 TDP2 (0.40) ALDH1A1SMN1; SMN2MAPTKDM4EMEN1
SCHEMBL10746773 0.65 ALDH1A1 (0.40) ALDH1A1NPC1RAB9ASMN1; SMN2LMNA
SCHEMBL6938561 0.64 ALDH1A1 (0.44) ALDH1A1POLBLMNAMAPTHTT
SCHEMBL9665346 0.63 USP2 (0.40) ALDH1A1MAPTKDM4EHTTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1628990-B1 NOVEL 14 AND 15 MEMBERED RING COMPOUNDS GLAXO GROUP LTD (GB) 2009-12-02 EP disclosed
US-20070141276-A1 Novel 14 and 15 membered ring compounds GLAXO GROUP LIMITED (GB) 2007-06-21 US disclosed
EP-1628990-A1 NOVEL 14 AND 15 MEMBERED RING COMPOUNDS GLAXO GROUP LIMITED (GB) 2006-03-01 EP disclosed
WO-2004101588-A1 NOVEL 14 AND 15 MEMBERED RING COMPOUNDS GLAXO GROUP LIMITED (GB) 2004-11-25 WO disclosed