SCHEMBL436008

SCHEMBL436008

COc1cccc2c(N)c(Cl)cnc12

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.44
ADRA1D P25100 2/20 0.44
ADRA1A P35348 2/20 0.44
ADRA1B P35368 2/20 0.44
HPGDS O60760 1/20 0.43
HAVCR2 Q8TDQ0 1/20 0.43
G6PD P11413 1/20 0.43
NQO2 P16083 1/20 0.43
MCHR1 Q99705 1/20 0.42
ATP4A P20648 1/20 0.42
ATP4B P51164 1/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP3A4 P08684 1/20 0.41
TDP1 Q9NUW8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL435849 0.81 HTR1A (0.44) HTR1AADRA1DADRA1AADRA1BHPGDS
SCHEMBL437559 0.80 HAVCR2 (0.40) HAVCR2KDM4ECYP3A4
SCHEMBL441707 0.79 HAVCR2 (0.63) HAVCR2KDM4EALDH1A1
SCHEMBL442075 0.78 HAVCR2 (0.46) HTR1AADRA1DADRA1AADRA1BHAVCR2
SCHEMBL441668 0.77 GAA (0.41) G6PDKDM4EALDH1A1
SCHEMBL439862 0.76 HAVCR2 (0.63) HAVCR2
SCHEMBL439519 0.75 DYRK1A (0.39) G6PDNQO2MCHR1KDM4EALDH1A1
SCHEMBL2178344 0.75 HTR1A (0.59) HTR1AADRA1DADRA1AADRA1BG6PD
SCHEMBL441422 0.75 HAVCR2 (0.46) HAVCR2
SCHEMBL437767 0.75 HAVCR2 (0.46) HAVCR2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed