SCHEMBL440416

SCHEMBL440416

Nc1c(Cl)cnc2c(F)cc(F)cc12

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CDK8 P49336 1/20 0.33
GSK3A P49840 1/20 0.33
GSK3B P49841 1/20 0.33
CDK9 P50750 1/20 0.33
CDK5 Q00535 1/20 0.33
DYRK1B Q9Y463 1/20 0.33
PIK3CD O00329 1/20 0.32
PIK3CB P42338 1/20 0.32
PDE10A Q9Y233 1/20 0.32
HAVCR2 Q8TDQ0 1/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
PKM P14618 1/20 0.30
RAB9A P51151 1/20 0.30
KMT2A Q03164 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
ALOX5AP P20292 1/20 0.30
FEN1 P39748 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL439456 0.79 CDK8 (0.33) CDK8GSK3AGSK3BCDK9CDK5
SCHEMBL441422 0.75 HAVCR2 (0.46) CDK9HAVCR2
SCHEMBL438931 0.73 HAVCR2 (0.49) CDK8GSK3AGSK3BCDK9CDK5
SCHEMBL440869 0.72 BCHE (0.46) HAVCR2ALDH1A1MAPT
SCHEMBL437520 0.71 AAK1 (0.34)
SCHEMBL442157 0.71 HAVCR2 (0.36) HAVCR2ALOX5APFEN1
SCHEMBL439645 0.71 ACHE (0.46)
4-Chloro-6,8-Difluoroquinoline SCHEMBL30225421 0.70 CDK8 (0.43) CDK8GSK3AGSK3BCDK9CDK5
4-Chloro-6,8-Difluoroquinoline SCHEMBL264453 0.70 CDK8 (0.43) CDK8GSK3AGSK3BCDK9CDK5
SCHEMBL441217 0.69 KDM4E (0.36) HAVCR2ALDH1A1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed