SCHEMBL441422

SCHEMBL441422

Nc1c(Cl)cnc2c(F)cccc12

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HAVCR2 Q8TDQ0 1/20 0.46
PARP1 P09874 1/20 0.41
NR4A2 P43354 2/20 0.40
GRM5 P41594 4/20 0.39
ACHE P22303 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.36
PIK3R2 O00459 1/20 0.35
CCNT1 O60563 1/20 0.34
CCNK O75909 1/20 0.34
CCNE1 P24864 1/20 0.34
CDK2 P24941 1/20 0.34
CDK7 P50613 1/20 0.34
CDK9 P50750 1/20 0.34
CCNH P51946 1/20 0.34
MNAT1 P51948 1/20 0.34
CDK12 Q9NYV4 1/20 0.34
TAAR1 Q96RJ0 1/20 0.34
PTGES O14684 1/20 0.34
JAK2 O60674 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL441707 0.83 HAVCR2 (0.63) HAVCR2PARP1NR4A2ACHESMN1; SMN2
SCHEMBL442157 0.79 HAVCR2 (0.36) HAVCR2
SCHEMBL435823 0.79 PARP1 (0.41) HAVCR2PARP1GRM5SMN1; SMN2
SCHEMBL442075 0.79 HAVCR2 (0.46) HAVCR2PARP1NR4A2ACHESMN1; SMN2
SCHEMBL437767 0.79 HAVCR2 (0.46) HAVCR2NR4A2ACHE
SCHEMBL18635471 0.79 PARP1 (0.41) HAVCR2PARP1GRM5PIK3R2
SCHEMBL437574 0.78 PARP1 (0.45) HAVCR2PARP1NR4A2CDK2
SCHEMBL23126271 0.75 PARP1 (0.41) HAVCR2PARP1GRM5SMN1; SMN2
SCHEMBL440416 0.75 CDK8 (0.33) HAVCR2CDK9
SCHEMBL16132381 0.75 GRM5 (0.40) PARP1GRM5PTGESJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed