SCHEMBL4411278

SCHEMBL4411278

COc1cccc(CNC(=O)c2cc(-c3cc(NC(=O)c4cc(C(C)(C)C)cc(C#N)c4OC)ccc3C)no2)c1OC

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.37
SCN9A Q15858 1/20 0.37
THRB P10828 1/20 0.37
ROCK2 O75116 2/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
ROCK1 Q13464 1/20 0.35
GAA P10253 2/20 0.35
NAMPT P43490 1/20 0.35
BRAF P15056 3/20 0.35
RAF1 P04049 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C19 P33261 1/20 0.34
MAOB P27338 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5593243 0.89 NPC1 (0.43) MAPTTHRBNPC1RAB9AGAA
SCHEMBL4565792 0.88 MAPT (0.41) MAPTTHRBNPC1RAB9ABRAF
SCHEMBL4411132 0.87 BRAF (0.38) MAPTTHRBBRAFRAF1CYP1A2
SCHEMBL4410129 0.86 MEN1 (0.44) MAPTNPC1RAB9ANAMPTBRAF
SCHEMBL4410261 0.85 NPC1 (0.39) MAPTTHRBNPC1RAB9AALDH1A1
SCHEMBL4420133 0.83 RAB9A (0.48) ROCK2NPC1RAB9AGAABRAF
SCHEMBL4410028 0.82 MAPT (0.38) MAPTTHRBBRAFRAF1KDM4E
SCHEMBL4414341 0.81 USP30 (0.40) NPC1RAB9ANAMPTBRAFRAF1
SCHEMBL4409883 0.81 MAPK14 (0.36) MAPTBRAFRAF1KDM4EALDH1A1
SCHEMBL5603582 0.80 MAPK14 (0.37) MAPTBRAFRAF1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035005-A2 THERAPY USING CYTOKINE INHIBITORS Kemia, INC. (US) 2009-03-18 EP disclosed
WO-2007146712-A2 THERAPY USING CYTOKINE INHIBITORS KEMIA, INC. (US) 2007-12-21 WO disclosed
WO-2007075896-A2 HETEROCYCLIC CYTOKINE INHIBITORS KEMIA, INC. (US) 2007-07-05 WO disclosed