SCHEMBL4403746

SCHEMBL4403746

O=C(NC1CCN(CCN2CCCCCC2)CC1)Oc1cc2c(OCc3ccoc3)cccc2[nH]1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36
CHRM3 P20309 1/20 0.36
SRD5A2 P31213 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
EPHX2 P34913 1/20 0.34
MCHR1 Q99705 3/20 0.34
KCNH2 Q12809 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
HTR4 Q13639 1/20 0.34
TMEM97 Q5BJF2 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34
CCR5 P51681 1/20 0.33
FAAH O00519 1/20 0.33
HRH2 P25021 1/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4409082 0.94 SRD5A2 (0.36) CHRM2CHRM1CHRM3SRD5A2MEN1
SCHEMBL4396602 0.89 SRD5A2 (0.47) SRD5A2MEN1KMT2ATMEM97FAAH
SCHEMBL4406699 0.89 KMT2A (0.34) CHRM2CHRM1CHRM3SRD5A2MEN1
SCHEMBL4396316 0.89 KMT2A (0.34) CHRM2CHRM1CHRM3SRD5A2MEN1
SCHEMBL4405956 0.89 FAAH (0.34) CHRM2CHRM1CHRM3SRD5A2MEN1
SCHEMBL914012 0.87 SRD5A2 (0.43) CHRM2CHRM1CHRM3SRD5A2MEN1
SCHEMBL4411388 0.87 CHRM2 (0.34) CHRM2CHRM1CHRM3SRD5A2MEN1
SCHEMBL4403443 0.86 MEN1 (0.35) MEN1KMT2AEPHX2MCHR1KCNH2
SCHEMBL4404430 0.84 HTR4 (0.37) EPHX2HRH3HTR4HTR2A
SCHEMBL4411341 0.84 HTR1A (0.34) SRD5A2MEN1KMT2AMCHR1CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720859-B1 CHEMOKINE RECEPTOR ANTAGONISTS NOVARTIS AG (CH) 2009-12-23 EP claimed