SCHEMBL4413087

SCHEMBL4413087

CCN(CC)C(=O)Cn1c(=O)oc2cc(Cl)ccc21

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.62
MAPT P10636 2/20 0.62
POLB P06746 1/20 0.62
LMNA P02545 3/20 0.55
CYP3A4 P08684 1/20 0.55
HPGD P15428 1/20 0.55
HSD17B10 Q99714 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
IDO1 P14902 3/20 0.50
PIK3CB P42338 1/20 0.49
KMT2A Q03164 3/20 0.48
MEN1 O00255 2/20 0.47
ALDH1A1 P00352 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4423635 0.88 TP53 (0.63) TP53MAPTPOLBLMNACYP3A4
SCHEMBL4414497 0.87 TP53 (0.61) TP53MAPTPOLBLMNACYP3A4
SCHEMBL4413124 0.86 TP53 (0.61) TP53MAPTPOLBLMNACYP3A4
SCHEMBL4423632 0.85 TSPO (0.57) TP53MAPTPOLBLMNACYP3A4
SCHEMBL4412637 0.81 MEN1 (0.63) POLBLMNACYP3A4HPGDKMT2A
SCHEMBL2978251 0.81 PIK3CB (0.58) TP53MAPTPOLBLMNACYP3A4
SCHEMBL4414360 0.80 HPGD (0.64) TP53MAPTPOLBLMNACYP3A4
SCHEMBL17830731 0.79 LMNA (0.61) TP53MAPTPOLBLMNACYP3A4
SCHEMBL4411764 0.79 TP53 (0.61) TP53MAPTPOLBLMNACYP3A4
SCHEMBL14044191 0.79 LMNA (0.59) TP53MAPTPOLBLMNACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8293775-B2 Benzoxazolone derivatives, processes for preparing them and their uses UCB PHARMA, S.A. (BE) 2012-10-23 US disclosed
EP-1756071-B1 BENZOXAZOLONE DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES UCB PHARMA SA (BE) 2009-08-26 EP disclosed
US-20070299118-A1 Benzoxazolone Derivatives, Processes For Preparing Them And Their Uses UCB, S.A. (BE) 2007-12-27 US disclosed
EP-1756071-A1 BENZOXAZOLONE DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES UCB, S.A. (BE) 2007-02-28 EP disclosed
WO-2005118561-A1 BENZOXAZOLONE DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES UCB, S.A. (BE) 2005-12-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070299118-A1 Benzoxazolone Derivatives, Processes For Preparing Them And Their Uses PARK7, SNCA, GABRA5 TP53 4794/4885MAPT 391/4885POLB 1027/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.