SCHEMBL435823

SCHEMBL435823

Nc1c(Br)cnc2c(F)cccc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.41
HAVCR2 Q8TDQ0 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CYP1A2 P05177 3/20 0.36
CYP3A4 P08684 3/20 0.36
CYP2C9 P11712 3/20 0.36
CYP2C19 P33261 3/20 0.36
TET2 Q6N021 1/20 0.36
GRM5 P41594 3/20 0.35
ALDH1A1 P00352 2/20 0.35
MEN1 O00255 1/20 0.35
APAF1 O14727 1/20 0.35
TDP2 O95551 1/20 0.35
MAPT P10636 1/20 0.35
CASP3 P42574 1/20 0.35
KMT2A Q03164 1/20 0.35
SENP8 Q96LD8 1/20 0.35
SENP7 Q9BQF6 1/20 0.35
SENP6 Q9GZR1 1/20 0.35
HKDC1 Q2TB90 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL442133 0.83 BACE1 (0.41) HAVCR2CYP1A2ALDH1A1MEN1APAF1
SCHEMBL441951 0.79 HAVCR2 (0.58) PARP1HAVCR2SMN1; SMN2CYP1A2ALDH1A1
SCHEMBL441701 0.79 ALDH1A1 (0.43) PARP1HAVCR2SMN1; SMN2CYP1A2ALDH1A1
SCHEMBL437507 0.79 MAP4K4 (0.35) TET2ALOX5APFEN1
SCHEMBL441422 0.79 HAVCR2 (0.46) PARP1HAVCR2SMN1; SMN2GRM5
SCHEMBL440370 0.78 PARP1 (0.45) PARP1
SCHEMBL23126271 0.75 PARP1 (0.41) PARP1HAVCR2SMN1; SMN2CYP3A4GRM5
SCHEMBL439456 0.75 CDK8 (0.33) TET2ALDH1A1MEN1MAPTKMT2A
SCHEMBL435849 0.75 HTR1A (0.44) CYP3A4
SCHEMBL437613 0.75 GABRA1 (0.41) PARP1HAVCR2ALDH1A1MEN1APAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed