SCHEMBL437574

SCHEMBL437574

Nc1c(Cl)cnc2c(C(F)(F)F)cccc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.45
HAVCR2 Q8TDQ0 1/20 0.43
NR1H2 P55055 14/20 0.42
NR1H3 Q13133 13/20 0.42
NCF1 P14598 1/20 0.39
NR4A2 P43354 1/20 0.37
DYRK3 O43781 1/20 0.36
PRKD3 O94806 1/20 0.36
MAP4K4 O95819 1/20 0.36
CDK1 P06493 1/20 0.36
CDK2 P24941 1/20 0.36
FLT4 P35916 1/20 0.36
CSNK1D P48730 1/20 0.36
CLK2 P49760 1/20 0.36
GSK3A P49840 1/20 0.36
GSK3B P49841 1/20 0.36
LIMK1 P53667 1/20 0.36
CSNK2A1 P68400 1/20 0.36
CDK5 Q00535 1/20 0.36
STK3 Q13188 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL440370 0.81 PARP1 (0.45) PARP1NR1H2NR1H3NCF1DYRK3
SCHEMBL441707 0.79 HAVCR2 (0.63) PARP1HAVCR2NR4A2PRKD3MAP4K4
SCHEMBL441422 0.78 HAVCR2 (0.46) PARP1HAVCR2NR4A2CDK2
SCHEMBL442075 0.78 HAVCR2 (0.46) PARP1HAVCR2NR4A2
SCHEMBL437559 0.77 HAVCR2 (0.40) HAVCR2NR4A2
SCHEMBL317787 0.75 NCF1 (0.51) PARP1NR1H2NR1H3NCF1NR4A2
SCHEMBL437767 0.75 HAVCR2 (0.46) HAVCR2NR4A2
SCHEMBL30880479 0.75 NCF1 (0.51) PARP1NR1H2NR1H3NCF1NR4A2
SCHEMBL436008 0.74 HTR1A (0.44) HAVCR2
SCHEMBL440440 0.74 HAVCR2 (0.47) PARP1HAVCR2NR4A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed