SCHEMBL4415834

SCHEMBL4415834

O=C1NC[C@](c2ccccc2)(C2CCCCC2)N1C1CCNCC1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 3/20 0.36
BACE2 Q9Y5Z0 3/20 0.36
APP P05067 1/20 0.36
CTSD P07339 1/20 0.36
CHRM3 P20309 2/20 0.35
CHRM2 P08172 1/20 0.35
GRIN1 Q05586 2/20 0.34
GRIN2A Q12879 2/20 0.34
GRIN2B Q13224 1/20 0.34
KDM4E B2RXH2 1/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
NSD3 Q9BZ95 1/20 0.33
SLC6A9 P48067 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4595948 1.00 BACE1 (0.36) BACE1BACE2APPCTSDCHRM3
SCHEMBL4596041 0.88 KDM4E (0.32) BACE1CHRM3KDM4ENSD3SLC6A9
SCHEMBL4597510 0.88 KDM4E (0.32) BACE1CHRM3KDM4ENSD3SLC6A9
SCHEMBL4596366 0.84 CHRM2 (0.37) BACE1CHRM3CHRM2SLC6A9
SCHEMBL4596721 0.84 CHRM2 (0.37) BACE1CHRM3CHRM2SLC6A9
SCHEMBL4597467 0.83 KDM4E (0.31) KDM4ENSD3
SCHEMBL4426327 0.80 SIGMAR1 (0.32) CHRM3GRIN1GRIN2AGRIN2B
SCHEMBL5179386 0.78 GRIN1 (0.38) CHRM3CHRM2GRIN1GRIN2AGRIN2B
SCHEMBL4610698 0.78 NSD3 (0.36) CHRM3CHRM2KDM4ENSD3
SCHEMBL4626507 0.78 NSD3 (0.36) CHRM3CHRM2KDM4ENSD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2088860-A1 CHEMOKINE RECEPTOR BINDING COMPOUNDS Genzyme Corporation (US) 2009-08-19 EP disclosed
WO-2008070758-A1 CHEMOKINE RECEPTOR BINDING COMPOUNDS GENZYME CORPORATION (US) 2008-06-12 WO disclosed
EP-1924265-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS Genzyme Corporation (US) 2008-05-28 EP disclosed
WO-2007022371-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS GENZYME CORPORATION (US) 2007-02-22 WO disclosed