SCHEMBL4596366

SCHEMBL4596366

O=C1NC[C@](c2cccc(Cl)c2)(C2CCCC2)N1C1CCNCC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.37
CHRM3 P20309 1/20 0.37
BACE1 P56817 3/20 0.36
DRD2 P14416 1/20 0.35
DPP4 P27487 3/20 0.35
DPP9 Q86TI2 3/20 0.35
DPP8 Q6V1X1 2/20 0.35
HTR2C P28335 2/20 0.35
HTR2B P41595 2/20 0.35
SLC6A4 P31645 2/20 0.35
HTR3E A5X5Y0 1/20 0.35
HTR3B O95264 1/20 0.35
TP53 P04637 1/20 0.35
CYP1A2 P05177 1/20 0.35
ADRB1 P08588 1/20 0.35
CYP3A4 P08684 1/20 0.35
HTR1A P08908 1/20 0.35
CYP2D6 P10635 1/20 0.35
THRB P10828 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596721 1.00 CHRM2 (0.37) CHRM2CHRM3BACE1DRD2DPP4
SCHEMBL4596506 0.90 DRD2 (0.34) BACE1DRD2DPP4DPP9DPP8
SCHEMBL4597256 0.90 DRD2 (0.34) BACE1DRD2DPP4DPP9DPP8
SCHEMBL4597579 0.86 DRD2 (0.33) DRD2DPP4DPP9DPP8HTR2C
SCHEMBL4415834 0.84 BACE1 (0.36) CHRM2CHRM3BACE1SLC6A9
SCHEMBL4595948 0.84 BACE1 (0.36) CHRM2CHRM3BACE1SLC6A9
SCHEMBL4597529 0.77 BACE1 (0.38) BACE1DRD2DPP4DPP9DPP8
SCHEMBL4596625 0.77 HTR2C (0.35) CHRM2CHRM3BACE1HTR2CHTR2B
SCHEMBL4598027 0.77 CHRNA1 (0.32) CHRM2CHRM3BACE1SLC6A4HTR6
SCHEMBL4597825 0.76 CHRM2 (0.39) CHRM2CHRM3DRD2DPP4DPP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924265-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS Genzyme Corporation (US) 2008-05-28 EP disclosed
WO-2007022371-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS GENZYME CORPORATION (US) 2007-02-22 WO disclosed