SCHEMBL4417546

SCHEMBL4417546

CC(C)CNC1CCC(CS(=O)(=O)c2ccccc2)(N2CC[C@H](Nc3ncnc4cc(C(C)(C)C)sc34)C2=O)CC1

nearest known ligand 0.32

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 10/20 0.32
CCR5 P51681 9/20 0.32
LPAR1 Q92633 1/20 0.31
LPAR2 Q9HBW0 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
ADRB2 P07550 1/20 0.30
ADRB1 P08588 1/20 0.30
ADRB3 P13945 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5027201 0.89 CCR2 (0.39) CCR2CCR5MEN1KMT2A
SCHEMBL4428634 0.89 TLR7 (0.32)
SCHEMBL4426062 0.84 CCR2 (0.37) CCR2CCR5
SCHEMBL4424140 0.84 IRAK4 (0.41) CCR2
SCHEMBL4426067 0.83 CNR1 (0.40) CCR2CCR5
SCHEMBL4551359 0.83 NSD2 (0.47)
SCHEMBL4417401 0.83 IRAK4 (0.39) CCR2CCR5
SCHEMBL4418746 0.83 CCR2 (0.49) CCR2CCR5
SCHEMBL4422907 0.82 PIK3CD (0.44) MEN1KMT2A
SCHEMBL4419993 0.82

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1606255-B1 CYCLIC DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL MYERS SQUIBB CO (US) 2009-11-11 EP claimed