SCHEMBL4417401

SCHEMBL4417401

CC(C)CNC1CCC(CS(=O)(=O)c2ccccc2)(N2CC[C@H](Nc3ncnc4ccc(F)cc34)C2=O)CC1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 1/20 0.39
CCR2 P41597 15/20 0.39
CCR5 P51681 14/20 0.38
CNR1 P21554 4/20 0.38
CNR2 P34972 3/20 0.38
CHRM2 P08172 1/20 0.37
CHRM4 P08173 1/20 0.37
CHRM1 P11229 1/20 0.37
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4424140 0.92 IRAK4 (0.41) IRAK4CCR2CNR1
SCHEMBL4418746 0.91 CCR2 (0.49) IRAK4CCR2CCR5CHRM2CHRM4
SCHEMBL4551359 0.89 NSD2 (0.47) IRAK4
SCHEMBL5030504 0.89 CCR2 (0.48) IRAK4CCR2CCR5CNR1CNR2
SCHEMBL4426067 0.87 CNR1 (0.40) CCR2CCR5CNR1CNR2
SCHEMBL4417824 0.85 FFAR2 (0.33) CCR2CCR5
SCHEMBL4424128 0.84 CCR2 (0.35) CCR2CCR5CNR1CNR2
SCHEMBL4422907 0.83 PIK3CD (0.44)
SCHEMBL4417546 0.83 CCR2 (0.32) CCR2CCR5
SCHEMBL4421314 0.82 CCR2 (0.38) CCR2CCR5CHRM2CHRM4CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1606255-B1 CYCLIC DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL MYERS SQUIBB CO (US) 2009-11-11 EP claimed