SCHEMBL4425554

SCHEMBL4425554

CNC(=O)OC(c1cn(S(=O)(=O)c2cnn(C)c2)c(-c2cccnc2F)c1F)C(C)(C)C

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
RORC P51449 4/20 0.33
SLC6A9 P48067 2/20 0.33
BRAF P15056 1/20 0.32
NAMPT P43490 2/20 0.31
GRIA2 P42262 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1837632 0.88 PTGS2 (0.30)
SCHEMBL1832698 0.86 RORC (0.32) RORCNAMPT
SCHEMBL2408490 0.86 HTR6 (0.35) GRIA2KCNH2
SCHEMBL1829458 0.86 RORC (0.32) RORCNAMPT
SCHEMBL2412509 0.85
SCHEMBL4425656 0.85 MET (0.39)
SCHEMBL4420426 0.85 KMT2A (0.33) RORC
SCHEMBL1835872 0.85 GRM4 (0.31)
SCHEMBL1831693 0.84
SCHEMBL2410027 0.83 NTRK1 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114917-A2 PYRROLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-11-11 EP disclosed
WO-2008108380-A2 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-12 WO disclosed