SCHEMBL2408490

SCHEMBL2408490

CNC(=O)OC(c1cn(S(=O)(=O)c2cccc(F)c2)c(-c2cccnc2F)c1F)C(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 16/20 0.35
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR7 P34969 1/20 0.33
ALDH1A1 P00352 1/20 0.32
DRD2 P14416 1/20 0.32
MET P08581 1/20 0.31
FGFR4 P22455 1/20 0.31
GRIA2 P42262 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4421014 0.93 HTR6 (0.34) HTR6HTR2AHTR2CHTR7DRD2
SCHEMBL4425656 0.93 MET (0.39) ALDH1A1MET
SCHEMBL2410874 0.92 NFE2L2 (0.35) HTR6HTR2AHTR2CHTR7ALDH1A1
SCHEMBL2410027 0.91 NTRK1 (0.31) ALDH1A1
SCHEMBL1832698 0.90 RORC (0.32)
SCHEMBL4425473 0.90 HTR6 (0.33) HTR6DRD2
SCHEMBL2414854 0.89 KDR (0.34) MET
SCHEMBL1837632 0.87 PTGS2 (0.30)
SCHEMBL1829458 0.86 RORC (0.32)
SCHEMBL2412509 0.86

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364979-A1 Pyrrole compounds Takeda Pharmaceutical Company Limited (JP) 2011-09-14 EP disclosed