SCHEMBL4428218

SCHEMBL4428218

CC(C)[Si](Oc1cc(Cl)c(C=O)c(Cl)c1)(C(C)C)C(C)C

nearest known ligand 0.36

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
KMT2A Q03164 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL282124 0.80 AKR1B1 (0.32) MEN1ALDH1A1KMT2ATDP1
SCHEMBL1076844 0.78 MEN1 (0.33) MEN1ALDH1A1KMT2ATDP1
SCHEMBL31725812 0.77
SCHEMBL1040963 0.76 ALDH1A3 (0.47) MEN1ALDH1A1KMT2ATDP1
SCHEMBL1250513 0.74 CA12 (0.39) MEN1ALDH1A1KMT2ATDP1
SCHEMBL15141254 0.74 DPP4 (0.36) ALDH1A1
SCHEMBL15145241 0.74 ALDH1A1 (0.38) ALDH1A1KMT2A
SCHEMBL4261649 0.73 IDO1 (0.35) MEN1ALDH1A1KMT2ATDP1
SCHEMBL18428478 0.73 ALDH1A1 (0.33) ALDH1A1
SCHEMBL207231 0.72 ERN1 (0.50) MEN1ALDH1A1KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025019825-A2 SUBSTITUTED 2-(3,5-DICHLORO-4-(4-HYDROXY-BENZYL)PHENOXY)ACETAMIDE DERIVATIVES BRII BIOSCIENCES, INC. (US) 2025-01-23 WO disclosed
WO-2023177667-A1 THYROID HORMONE RECEPTOR AGONISTS BRII BIOSCIENCES, INC. (US) 2023-09-21 WO disclosed
EP-1678163-B1 NOVEL IMIDAZOLE DERIVATIVES AND THEIR USE AS PHARMACEUTICAL AGENTS HOFFMANN LA ROCHE (CH) 2009-01-07 EP disclosed
EP-1499577-B1 2-(2,6-DICHLOROPHENYL)-DIARYLIMIDAZOLES HOFFMANN LA ROCHE (CH) 2007-05-30 EP disclosed
US-7169781-B2 Imidazole derivatives and their use as pharmaceutical agents HOFFMANN-LA ROCHE INC. (US) 2007-01-30 US disclosed
US-7144889-B2 Triarylimidazoles HOFFMAN-LA ROCHE INC. (US) 2006-12-05 US disclosed
EP-1678163-A1 NOVEL IMIDAZOLE DERIVATIVES AND THEIR USE AS PHARMACEUTICAL AGENTS F. HOFFMANN-LA ROCHE AG (CH) 2006-07-12 EP disclosed
EP-1675848-A1 NOVEL TRIARYLIMIDAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2006-07-05 EP disclosed
US-6946471-B2 2-(2,6-Dichlorophenyl)-Diarylimidazoles HOFFMANN-LA ROCHE INC. (US) 2005-09-20 US disclosed
US-20050113342-A1 Novel imidazole derivatives and their use as pharmaceutical agents HOFFMANN-LA ROCHE INC. 2005-05-26 US disclosed
WO-2005040153-A1 NOVEL TRIARYLIMIDAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2005-05-06 WO disclosed
WO-2005040154-A1 NOVEL IMIDAZOLE DERIVATIVES AND THEIR USE AS PHARMACEUTICAL AGENTS F. HOFFMANN-LA ROCHE AG (CH) 2005-05-06 WO disclosed
US-20050085473-A1 Novel triarylimidazoles HOFFMANN-LA ROCHE INC. 2005-04-21 US disclosed
EP-1499577-A1 2-(2,6-DICHLOROPHENYL)-DIARYLIMIDAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2005-01-26 EP disclosed
US-20040214874-A1 2-(2,6-Dichlorophenyl)-Diarylimidazoles BRANDT MICHAEL 2004-10-28 US disclosed
US-6790852-B2 HETEROCYCLIC NITROGEN COMPOUNDS SUCH AS 2-(2,6-DICHLOROPHENYL) -4-(3-BROMOPHENYL)-5-(2-(3- HYDROXYPROPYLAMINO)PYRIMIDIN-4-YL) -N-H-IMIDAZOLE, USED AS TYROSINE KINASE INHIBITORS; ANTICARCINOGENIC OR ANTITUMOR AGENTS HOFFMANN-LA ROCHE INC. 2004-09-14 US disclosed
US-20030199691-A1 2-(2,6-dichlorophenyl)-diarylimidazoles F. HOFFMANN-LA ROCHE AG (CH) 2003-10-23 US disclosed
WO-2003087026-A1 2-(2,6-DICHLOROPHENYL)-DIARYLIMIDAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2003-10-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050085473-A1 Novel triarylimidazoles AURKAIP1, GLS2, GOT2 MEN1 1927/4885ALDH1A1 409/4885KMT2A 2396/4885
US-20050113342-A1 Novel imidazole derivatives and their use as pharmaceutical agents TUBB6, ABCB1, SDHA MEN1 608/4885ALDH1A1 265/4885KMT2A 3524/4885
US-20030199691-A1 2-(2,6-dichlorophenyl)-diarylimidazoles CYP2D6, CYP2F1, CYP1A2 MEN1 1726/4885ALDH1A1 115/4885KMT2A 933/4885
US-20040214874-A1 2-(2,6-Dichlorophenyl)-Diarylimidazoles CYP2D6, CYP1A2, CYP2F1 MEN1 1918/4885ALDH1A1 89/4885KMT2A 858/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.