SCHEMBL282124

SCHEMBL282124

Cc1cc(O[Si](C(C)C)(C(C)C)C(C)C)cc(C)c1C=O

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 5/20 0.32
ALB P02768 1/20 0.31
KDM4E B2RXH2 1/20 0.30
MEN1 O00255 1/20 0.30
NPC1 O15118 1/20 0.30
USP2 O75604 1/20 0.30
LDHA P00338 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
ESR1 P03372 1/20 0.30
TP53 P04637 1/20 0.30
CYP1A2 P05177 1/20 0.30
POLB P06746 1/20 0.30
LDHB P07195 1/20 0.30
CYP3A4 P08684 1/20 0.30
GAA P10253 1/20 0.30
AR P10275 1/20 0.30
BCL2 P10415 1/20 0.30
CYP2D6 P10635 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4428218 0.80 MEN1 (0.36) MEN1ALDH1A1KMT2ATDP1
SCHEMBL5379601 0.77 ALDH1A1 (0.39) KDM4EMEN1NPC1ALDH1A1CYP1A2
SCHEMBL28985344 0.77 HPGD (0.40) AKR1B1ALDH1A1LMNAMAPTHPGD
SCHEMBL1620823 0.75 ALDH1A3 (0.34) KDM4ENPSR1
SCHEMBL18428478 0.75 ALDH1A1 (0.33) ALDH1A1
SCHEMBL282196 0.75 ALDH1A1 (0.41) ALDH1A1LMNAMAPTHPGD
SCHEMBL19265771 0.75 ALDH1A3 (0.48) AKR1B1ALBKDM4EMEN1NPC1
SCHEMBL282712 0.75 ALDH1A1 (0.41) ALDH1A1TP53POLBCYP3A4TDP1
SCHEMBL1251338 0.73 CA12 (0.40)
SCHEMBL1619909 0.71 CYP1A1 (0.44) KDM4EMEN1NPC1USP2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 28 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115819288-B Nitrile oxide, difunctional nitrile oxide and preparation method thereof 西安近代化学研究所 2024-05-28 CN claimed
CN-115819288-A Nitrile oxide, bifunctional nitrile oxide and preparation method thereof 西安近代化学研究所 2023-03-21 CN claimed
EP-4662219-A2 PRODRUGS OF THYROID HORMONE ANALOGS, METHODS OF MAKING AND METHODS OF USING THEREOF ASCLETIS PHARMA (CHINA) CO., LIMITED (HK) 2025-12-17 EP disclosed
EP-4644357-A1 COMPOUND USEFUL AS THYROID HORMONE RECEPTOR B-SELECTIVE THYROID HORMONE ANALOG NATIONAL UNIVERSITY CORPORATION TOKAI NATIONAL HIGHER EDUCATION AND RESEARCH SYSTEM (JP) 2025-11-05 EP disclosed
US-20240294561-A1 Prodrugs of Thyroid Hormone Analogs, Methods of Making and Methods of Using Thereof ASCLETIS PHARMA (CHINA) CO., LIMITED (CN) 2024-09-05 US disclosed
WO-2024167961-A2 PRODRUGS OF THYROID HORMONE ANALOGS, METHODS OF MAKING AND METHODS OF USING THEREOF GANNEX, LLC (US) 2024-08-15 WO disclosed
WO-2024143235-A1 COMPOUND USEFUL AS THYROID HORMONE RECEPTOR β-SELECTIVE THYROID HORMONE ANALOG 国立大学法人東海国立大学機構 2024-07-04 WO disclosed
CN-115819288-B Nitrile oxide, difunctional nitrile oxide and preparation method thereof 西安近代化学研究所 2024-05-28 CN disclosed
CN-112300211-B Compound serving as thyroid hormone beta receptor agonist and application thereof 广东东阳光药业股份有限公司 2023-12-08 CN disclosed
US-20230339993-A1 PREPARATION METHOD OF A CYCLIC PHOSPHONATE COMPOUND GANNEX PHARMA CO., LTD. (CN) 2023-10-26 US disclosed
US-11725019-B2 Preparation method of a cyclic phosphonate compound GANNEX PHARMA CO LTD. (CN) 2023-08-15 US disclosed
EP-1689383-A4 NOVEL PHOSPHORUS-CONTAINING THYROMIMETICS METABASIS THERAPEUTICS INC (US) 2009-02-18 EP disclosed
US-20090028925-A1 Novel Phosphinic Acid-Containing Thyromimetics METABASIS THERAPEUTICS, INC. 2009-01-29 US disclosed
EP-1891080-A2 NOVEL PHOSPHORUS-CONTAINING THYROMIMETICS Metabasis Therapeutics, Inc. (US) 2008-02-27 EP disclosed
EP-1890768-A2 NOVEL PHOSPHINIC ACID-CONTAINING THYROMIMETICS Metabasis Therapeutics, Inc. (US) 2008-02-27 EP disclosed
WO-2006128056-A2 NOVEL PHOSPHINIC ACID-CONTAINING THYROMIMETICS METABASIS THERAPEUTICS, INC. (US) 2006-11-30 WO disclosed
WO-2006128055-A2 NOVEL PHOSPHORUS-CONTAINING THYROMIMETICS METABASIS THERAPEUTICS, INC. (US) 2006-11-30 WO disclosed
EP-1689383-A2 NOVEL PHOSPHORUS-CONTAINING THYROMIMETICS Metabasis Therapeutics, Inc. (US) 2006-08-16 EP disclosed
US-20060046980-A1 Novel phosphorus-containing thyromimetics METABASIS THERAPEUTICS, INC. 2006-03-02 US disclosed
WO-2005051298-A2 NOVEL PHOSPHORUS-CONTAINING THYROMIMETICS METABASIS THERAPEUTICS, INC. (US) 2005-06-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240294561-A1 Prodrugs of Thyroid Hormone Analogs, Methods of Making and Methods of Using Thereof THRB, THRA, TSHR AKR1B1 397/4885ALB 4425/4885KDM4E 3558/4885
US-11725019-B2 Preparation method of a cyclic phosphonate compound PHOSPHO1, PPIP5K2, PNKP AKR1B1 1355/4885ALB 2930/4885KDM4E 4335/4885
US-20060046980-A1 Novel phosphorus-containing thyromimetics PYGL, THRA, THOP1 AKR1B1 1452/4885ALB 1996/4885KDM4E 4102/4885
US-20230339993-A1 PREPARATION METHOD OF A CYCLIC PHOSPHONATE COMPOUND PHOSPHO1, PPIP5K2, PNKP AKR1B1 1355/4885ALB 2930/4885KDM4E 4335/4885
US-20090028925-A1 Novel Phosphinic Acid-Containing Thyromimetics PYGL, PHOSPHO1, LIPE AKR1B1 1741/4885ALB 1305/4885KDM4E 4083/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.