SCHEMBL4437699

SCHEMBL4437699

COC(=O)c1ccc(Cc2ccccc2-c2ccc(F)cc2)[nH]c1=O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 4/20 0.55
SLC6A4 P31645 3/20 0.55
KDM4E B2RXH2 2/20 0.43
GLA P06280 1/20 0.43
GAA P10253 1/20 0.43
LIPG Q9Y5X9 1/20 0.41
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40
NPC1 O15118 1/20 0.40
CASP3 P42574 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
SENP8 Q96LD8 1/20 0.40
SENP7 Q9BQF6 1/20 0.40
SENP6 Q9GZR1 1/20 0.40
PTGDR2 Q9Y5Y4 2/20 0.40
SLC6A2 P23975 1/20 0.39
CYP1A2 P05177 3/20 0.39
ALDH1A1 P00352 2/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4438513 0.91 KDM4E (0.47) SLC6A3SLC6A4KDM4EGLAGAA
SCHEMBL4430819 0.86 BRS3 (0.46) SLC6A3SLC6A4KDM4ELIPGPTGDR2
SCHEMBL4431012 0.85 SLC6A3 (0.58) SLC6A3SLC6A4KDM4EGLAGAA
SCHEMBL4439655 0.81 MAPK8 (0.45) KDM4EGLAGAAPDE3BPDE3A
SCHEMBL3913842 0.80 KDM4E (0.51) SLC6A3SLC6A4KDM4EGLAGAA
SCHEMBL4431808 0.79 KDM4E (0.50) KDM4EGLAGAAPDE3BPDE3A
SCHEMBL4426834 0.78 ALDH1A1 (0.54) KDM4EGLAGAAPDE3BPDE3A
SCHEMBL4433888 0.76 KDM4E (0.53) KDM4EGAASMN1; SMN2ALDH1A1BRS3
SCHEMBL4432962 0.76 MDM2 (0.42) KDM4EGAAPDE3BPDE3ANPC1
SCHEMBL4426842 0.76 KDM4E (0.49) SLC6A3SLC6A4KDM4EGLAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125739-A1 MODULATORS OF C3A RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. (US) 2009-12-02 EP disclosed
WO-2008079371-A1 MODULATORS OF C3A RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-07-03 WO disclosed