SCHEMBL4444902

SCHEMBL4444902

O=CC(O)C1(c2ccsc2)CC1

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 1/20 0.33
SLC6A2 P23975 3/20 0.32
SLC6A4 P31645 3/20 0.32
SLC6A3 Q01959 1/20 0.32
HCAR3 P49019 1/20 0.31
HCAR2 Q8TDS4 1/20 0.31
CES2 O00748 1/20 0.31
CES1 P23141 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4438204 0.71 CYP2A6 (0.34) SLC6A3
SCHEMBL4437241 0.69 SLC6A3 (0.45) CHRM1SLC6A2SLC6A4SLC6A3
SCHEMBL27083166 0.68 CHRM1 (0.34) CHRM1SLC6A2SLC6A4SLC6A3HCAR3
SCHEMBL4446504 0.68 MAOA (0.39) SLC6A2SLC6A4SLC6A3CES2CES1
SCHEMBL27082164 0.66 CHRM1 (0.33) CHRM1SLC6A2SLC6A4SLC6A3HCAR3
SCHEMBL1310070 0.65
SCHEMBL4440469 0.65 SLC6A4 (0.50) SLC6A2SLC6A4SLC6A3
SCHEMBL28018276 0.64 CES2 (0.40) CHRM1SLC6A2SLC6A4SLC6A3HCAR3
SCHEMBL27082374 0.64 KCNA3 (0.36) CHRM1SLC6A2SLC6A4SLC6A3
SCHEMBL4435076 0.64 KDM1A (0.44) SLC6A2SLC6A4SLC6A3CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2134692-A2 QUINOLINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM FOR SELECTIN INHIBITION Wyeth a Corporation of the State of Delaware (US) 2009-12-23 EP disclosed
WO-2008121817-A2 QUINOLINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM FOR SELECTIN INHIBITION WYETH (US) 2008-10-09 WO disclosed