SCHEMBL4447858

SCHEMBL4447858

CCOC(=O)NCC(O)c1cccc(C(F)(F)F)c1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PNMT P11086 1/20 0.51
THRB P10828 1/20 0.49
NPC1 O15118 3/20 0.49
RAB9A P51151 3/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
LMNA P02545 1/20 0.49
POLB P06746 2/20 0.45
KMT2A Q03164 2/20 0.45
CES2 O00748 1/20 0.45
ALDH1A1 P00352 3/20 0.44
GAA P10253 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
KDM4E B2RXH2 1/20 0.44
MAPT P10636 1/20 0.44
HTT P42858 1/20 0.44
MEN1 O00255 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10217175 0.86 THRB (0.48) PNMTTHRBSMN1; SMN2POLBKMT2A
SCHEMBL4436210 0.86 THRB (0.48) PNMTTHRBSMN1; SMN2POLBKMT2A
SCHEMBL257275 0.85 PNMT (0.51) PNMTCES2ALDH1A1L3MBTL1
SCHEMBL19265132 0.84 THRB (0.47) THRBSMN1; SMN2POLBKMT2AALDH1A1
SCHEMBL4440894 0.84 PNMT (0.59) PNMTNPC1RAB9ASMN1; SMN2POLB
SCHEMBL4437771 0.84 PNMT (0.59) PNMTNPC1RAB9ASMN1; SMN2POLB
SCHEMBL10217045 0.82 FAAH (0.45) THRBPOLBKMT2AALDH1A1GAA
SCHEMBL10441979 0.80 SMN1; SMN2 (0.72) NPC1RAB9ASMN1; SMN2LMNAPOLB
SCHEMBL5704283 0.80 SMN1; SMN2 (0.72) NPC1RAB9ASMN1; SMN2LMNAPOLB
SCHEMBL8062422 0.80 SMN1; SMN2 (0.72) NPC1RAB9ASMN1; SMN2LMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121598-A2 COMPOUNDS AND COMPOSITIONS AS INHIBITORS OF CANNABINOID RECEPTOR 1 ACTIVITY IRM LLC (BM) 2009-11-25 EP disclosed
WO-2008076754-A2 COMPOUNDS AND COMPOSITIONS AS INHIBITORS OF CANNABINOID RECEPTOR 1 ACTIVITY IRM LLC (BM) 2008-06-26 WO disclosed