SCHEMBL4465846

SCHEMBL4465846

CS(=O)(=O)OCC=CCOS(C)(=O)=O

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
USP2 O75604 2/20 0.48
TSHR P16473 2/20 0.48
ALDH1A1 P00352 2/20 0.48
KDM4E B2RXH2 1/20 0.48
LMNA P02545 1/20 0.48
MMP9 P14780 1/20 0.48
ALOX15 P16050 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6118063 1.00 USP2 (0.48) USP2TSHRALDH1A1KDM4ELMNA
SCHEMBL4465842 1.00 USP2 (0.48) USP2TSHRALDH1A1KDM4ELMNA
SCHEMBL9675619 0.89 USP2 (0.40) USP2TSHRALDH1A1KDM4ELMNA
SCHEMBL4361309 0.89 USP2 (0.40) USP2TSHRALDH1A1KDM4ELMNA
SCHEMBL4361313 0.89 USP2 (0.40) USP2TSHRALDH1A1KDM4ELMNA
SCHEMBL7480571 0.86
SCHEMBL7480573 0.86
SCHEMBL7804173 0.85 ALDH1A1 (0.37) USP2TSHRALDH1A1KDM4ELMNA
SCHEMBL2167533 0.85 KDM4E (0.37) USP2TSHRALDH1A1KDM4ELMNA
SCHEMBL2167535 0.85 KDM4E (0.37) USP2TSHRALDH1A1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 46 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240229026-A1 CHIRAL CONTROL WAVE LIFE SCIENCES LTD. (SG) 2024-07-11 US disclosed
EP-4219516-A2 CHIRAL CONTROL Wave Life Sciences Ltd. (SG) 2023-08-02 EP disclosed
US-11643657-B2 Chiral control WAVE LIFE SCIENCES LTD. (SG) 2023-05-09 US disclosed
EP-2872147-B1 METHOD FOR MAKING CHIRAL OLIGONUCLEOTIDES WAVE LIFE SCIENCES LTD (SG) 2022-12-21 EP disclosed
US-11114693-B2 Electrolytic solution for nonaqueous electrolytic solution secondary batteries and nonaqueous electrolytic solution secondary battery CENTRAL GLASS COMPANY, LTD. (JP) 2021-09-07 US disclosed
US-20210130821-A1 CHIRAL CONTROL WAVE LIFE SCIENCES LTD. (SG) 2021-05-06 US disclosed
CN-107851847-B Nonaqueous electrolyte solution and nonaqueous electrolyte battery using same 中央硝子株式会社 2020-12-18 CN disclosed
EP-3333962-B1 ELECTROLYTIC SOLUTION FOR NONAQUEOUS ELECTROLYTIC SOLUTION SECONDARY BATTERIES AND NONAQUEOUS ELECTROLYTIC SOLUTION SECONDARY BATTERY CENTRAL GLASS CO LTD (JP) 2020-10-07 EP disclosed
US-20200212485-A1 Non-Aqueous Electrolyte Solution and Non-Aqueous Electrolyte Battery in Which Same Is Used CENTRAL GLASS COMPANY, LIMITED (JP) 2020-07-02 US disclosed
US-10590413-B2 Chiral control WAVE LIFE SCIENCES LTD. (SG) 2020-03-17 US disclosed
WO-2009090548-A2 3-AZABICYCLO [3.1.0] HEXANE DERIVATIVES AS VANILLOID RECEPTOR LIGANDS GLENMARK PHARMACEUTICALS, S.A. (US) 2009-07-23 WO disclosed
WO-2008010061-A2 3-AZABICYCLO [3.1.0] HEXANE VANILLOID RECEPTOR LIGANDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM, AND PROCESSES FOR THEIR PREPARATION GLENMARK PHARMACEUTICALS S.A. (US) 2008-01-24 WO disclosed
EP-1375496-B1 N-ARYL-SUBSTITUTED CYCLIC AMINE DERIVATIVE AND MEDICINE CONTAINING THE SAME AS ACTIVE INGREDIENT EISAI R&D MAN CO LTD (JP) 2007-07-04 EP disclosed
US-7112593-B2 N-aryl-substituted cyclic amine derivative and medicine containing the same as active ingredient EISAI CO., LTD. (JP) 2006-09-26 US disclosed
US-20060079533-A1 Methods of treating alzheimer's disease NIEMAN JAMES A 2006-04-13 US disclosed
US-20040072830-A1 N-aryl-substituted cyclic amine derivative and medicine containing the same as active ingredient EISAI R&D MANAGEMENT CO., LTD. (JP) 2004-04-15 US disclosed
EP-1375496-A1 N-ARYL-SUBSTITUTED CYCLIC AMINE DERIVATIVE AND MEDICINE CONTAINING THE SAME AS ACTIVE INGREDIENT Eisai Co., Ltd. (JP) 2004-01-02 EP disclosed
WO-2002076440-A2 METHODS OF TREATING ALZHEIMER'S DISEASE WITH PIPERIDIN DERIVATES ELAN PHARMACEUTICALS, INC. (US) 2002-10-03 WO disclosed
US-6150526-A Piperidine derivative having renin inhibiting activity HOFFMANN-LA ROCHE INC. (US) 2000-11-21 US disclosed
US-6051712-A PREVENTION OF HIGH BLOOD PRESSURE AND CARDIAC INSUFFICIENCY, AS WELL AS GLAUCOMA, CARDIAC INFARCT, KIDNEY INSUFFICIENCY AND RESTENOSIS HOFFMANN-LA ROCHE INC. (US) 2000-04-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210130821-A1 CHIRAL CONTROL RNGTT, POLI, NSUN3 USP2 3936/4885TSHR 3259/4885ALDH1A1 2867/4885
US-20040072830-A1 N-aryl-substituted cyclic amine derivative and medicine containing the same as active ingredient COASY, HCCS, SQLE USP2 3445/4885TSHR 3428/4885ALDH1A1 1799/4885
US-11114693-B2 Electrolytic solution for nonaqueous electrolytic solution secondary batteries and nonaqueous electrolytic solution secondary battery ESPL1, TST, PEF1 USP2 4743/4885TSHR 4303/4885ALDH1A1 1379/4885
US-20240229026-A1 CHIRAL CONTROL RNGTT, POLI, NSUN3 USP2 3936/4885TSHR 3259/4885ALDH1A1 2867/4885
US-20200212485-A1 Non-Aqueous Electrolyte Solution and Non-Aqueous Electrolyte Battery in Which Same Is Used SLC9A1, TST, CA1 USP2 4694/4885TSHR 4390/4885ALDH1A1 891/4885
US-11643657-B2 Chiral control RNGTT, POLI, NSUN3 USP2 3936/4885TSHR 3259/4885ALDH1A1 2867/4885
US-10590413-B2 Chiral control RNGTT, POLI, NSUN3 USP2 3936/4885TSHR 3259/4885ALDH1A1 2867/4885
US-20060079533-A1 Methods of treating alzheimer's disease BACE1, PSEN1, PSEN2 USP2 1490/4885TSHR 3417/4885ALDH1A1 2504/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.