Betamipron

Betamipron

SCHEMBL4498475

O=C(O)CCNC(=O)c1ccccc1.c1ccccc1

nearest known ligand 0.76

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 1/20 0.70
CTSG P08311 1/20 0.70
CTRB1 P17538 1/20 0.70
CMA1 P23946 1/20 0.70
GAA P10253 1/20 0.63
CA1 P00915 1/20 0.62
CA2 P00918 1/20 0.62
SMN1; SMN2 Q16637 4/20 0.61
LMNA P02545 2/20 0.61
MAPK1 P28482 1/20 0.61
POLB P06746 1/20 0.61
NPC1 O15118 4/20 0.59
RAB9A P51151 4/20 0.59
EPHX2 P34913 1/20 0.59
HDAC3 O15379 3/20 0.58
HDAC4 P56524 3/20 0.58
HDAC1 Q13547 3/20 0.58
HDAC7 Q8WUI4 3/20 0.58
HDAC2 Q92769 3/20 0.58
HDAC10 Q969S8 3/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Betamipron SCHEMBL605899 1.00 PRSS1 (0.70) PRSS1CTSGCTRB1CMA1GAA
SCHEMBL9717434 0.91 MAPK1 (0.71) PRSS1CTSGCTRB1CMA1GAA
SCHEMBL2033165 0.88 MAPK1 (0.73) PRSS1CTSGCTRB1CMA1GAA
SCHEMBL9717417 0.88 ITGB3 (0.65) PRSS1CTSGCTRB1CMA1GAA
SCHEMBL9829615 0.87 GAA (0.57) PRSS1CTSGCTRB1CMA1GAA
SCHEMBL3192014 0.87 LMNA (0.77) PRSS1CTSGCTRB1CMA1GAA
Betamipron SCHEMBL28084518 0.87 NPC1 (0.73) PRSS1CTSGCTRB1CMA1SMN1; SMN2
SCHEMBL950223 0.86 MAPK1 (0.83) PRSS1CTSGCTRB1CMA1GAA
SCHEMBL2324530 0.86 PRSS1 (0.64) PRSS1CTSGCTRB1CMA1GAA
SCHEMBL5592824 0.86 PRSS1 (0.68) PRSS1CTSGCTRB1CMA1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7517858-B1 Prodrugs of pharmaceuticals with improved bioavailability THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2009-04-14 US disclosed
EP-0837630-A4 PRODRUGS OF PHARMACEUTICALS WITH IMPROVED BIOAVAILABILITY UNIV CALIFORNIA (US) 1998-11-25 EP disclosed
EP-0837630-A1 PRODRUGS OF PHARMACEUTICALS WITH IMPROVED BIOAVAILABILITY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1998-04-29 EP disclosed
WO-1996039831-A1 PRODRUGS OF PHARMACEUTICALS WITH IMPROVED BIOAVAILABILITY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1996-12-19 WO disclosed