SCHEMBL4518320

SCHEMBL4518320

O=C(O)C(=O)c1cccc(F)c1

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.79
CES1 P23141 2/20 0.79
PARP1 P09874 1/20 0.61
HDAC1 Q13547 1/20 0.57
HDAC6 Q9UBN7 1/20 0.57
MEN1 O00255 4/20 0.51
KMT2A Q03164 4/20 0.51
KCNK3 O14649 1/20 0.51
NPC1 O15118 3/20 0.50
RAB9A P51151 2/20 0.50
HPGD P15428 2/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
PLA2G7 Q13093 1/20 0.50
PKM P14618 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
GAA P10253 1/20 0.46
KAT6A Q92794 1/20 0.46
ESR1 P03372 1/20 0.46
ESR2 Q92731 1/20 0.46
GPR52 Q9Y2T5 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15180847 1.00 CES2 (0.79) CES2CES1PARP1HDAC1HDAC6
SCHEMBL3169331 0.89 CES2 (1.00) CES2CES1PARP1HDAC1HDAC6
SCHEMBL7604854 0.84 L3MBTL1 (0.56) CES2CES1L3MBTL1PKMTSHR
SCHEMBL29665004 0.82 CES2 (0.71) CES2CES1PARP1HDAC1HDAC6
SCHEMBL28396 0.82 CES2 (0.71) CES2CES1PARP1HDAC1HDAC6
SCHEMBL13950378 0.82 CES2 (0.71) CES2CES1PARP1HDAC1HDAC6
SCHEMBL28788147 0.81 CES2 (0.63) CES2CES1PARP1HDAC1HDAC6
SCHEMBL29019528 0.81 CES2 (0.63) CES2CES1PARP1HDAC1HDAC6
SCHEMBL22718375 0.81 CES2 (0.76) CES2CES1PARP1HDAC1HDAC6
SCHEMBL3650973 0.81 CES2 (0.76) CES2CES1PARP1HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 36 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109575032-A The method of level-one amine guiding building 6- (3- fluorophenyl) indoles simultaneously [1,2-a] quinoxaline 桂林理工大学 2019-04-05 CN claimed
EP-0975584-B1 SYNTHESIS AND USE OF ALPHA-KETOAMIDE DERIVATIVES AND ARRAYS ARQULE INC (US) 2002-09-25 EP claimed
JP-60215647-A None JP disclosed
EP-4095162-A1 APPLICATION OF AND PREPARATION METHOD FOR CATIONIC POLYMER MODIFIED BY FLUORINE-CONTAINING COMPOUND AS DRUG CARRIER Soochow University (CN) 2022-11-30 EP disclosed
CN-114956933-A Marker containing isotope oxygen atom and preparation method and application thereof 清华大学 2022-08-30 CN disclosed
CN-109575032-A The method of level-one amine guiding building 6- (3- fluorophenyl) indoles simultaneously [1,2-a] quinoxaline 桂林理工大学 2019-04-05 CN disclosed
CN-109575032-A The method of level-one amine guiding building 6- (3- fluorophenyl) indoles simultaneously [1,2-a] quinoxaline 桂林理工大学 2019-04-05 CN disclosed
CN-108017635-A A kind of method of successive reaction synthesizing aryl benzoquinolizine ketone compounds 黑龙江大学 2018-05-11 CN disclosed
US-20170296681-A1 COMPOSITIONS AND METHODS FOR IMAGING THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2017-10-19 US disclosed
EP-2661428-B1 QUINOXALINES AND AZA-QUINOXALINES AS CRTH2 RECEPTOR MODULATORS MERCK SHARP & DOHME (US) 2017-06-07 EP disclosed
EP-2661428-B1 QUINOXALINES AND AZA-QUINOXALINES AS CRTH2 RECEPTOR MODULATORS MERCK SHARP & DOHME (US) 2017-06-07 EP disclosed
WO-2012087861-A1 QUINOXALINES AND AZA-QUINOXALINES AS CRTH2 RECEPTOR MODULATORS MERCK SHARP & DOHME CORP. (US) 2012-06-28 WO disclosed
US-20090306062-A1 2,5-Disubstituted Piperidines NOVARTIS AG (CH) 2009-12-10 US disclosed
CN-1188471-A 1,4-disubstituted piepridine derivatives BANYU PHARMA CO LTD (JP) 1998-07-22 CN disclosed
US-5334726-A Controlling weeds ROHM AND HAAS COMPANY (US) 1994-08-02 US disclosed
US-5120347-A Pre and postemergence ROHM AND HAAS COMPANY (US) 1992-06-09 US disclosed
US-4801708-A FOR AGRICULTURAL USE CIBA-GEIGY CORPORATION (US) 1989-01-31 US disclosed
EP-0150677-B1 HERBICIDAL AND INSECTICIDAL TRIAZINONES CIBA-GEIGY AG (CH) 1989-01-18 EP disclosed
JP-S60215647-A PREPARATION OF AROMATIC ALPHA-HYDROXY ACID AJINOMOTO CO INC 1985-10-29 JP disclosed
EP-0150677-A1 Herbicidal and insecticidal triazinones CIBA-GEIGY AG (CH) 1985-08-07 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170296681-A1 COMPOSITIONS AND METHODS FOR IMAGING GPX4, PRDX5, PRDX2 CES2 1320/4885CES1 1166/4885PARP1 3012/4885
US-20090306062-A1 2,5-Disubstituted Piperidines REN, AGTR1, AGTR2 CES2 247/4885CES1 328/4885PARP1 1566/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.