SCHEMBL4527677

SCHEMBL4527677

Nc1c(Cc2ccccc2)c(C2CCCC2)c(Cc2ccccc2)c(N)c1C1CCCC1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.38
GABRG2 P18507 1/20 0.38
GABRB3 P28472 1/20 0.38
CCR2 P41597 1/20 0.37
CALM1 P0DP23 1/20 0.37
NR3C1 P04150 2/20 0.35
NOS3 P29474 1/20 0.35
NOS1 P29475 1/20 0.35
NOS2 P35228 1/20 0.35
CYP19A1 P11511 1/20 0.35
RAB9A P51151 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
TNK2 Q07912 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1499291 0.98 GABRA1 (0.38) GABRA1GABRG2GABRB3CCR2CALM1
SCHEMBL1499436 0.88 GABRA1 (0.36) GABRA1GABRG2GABRB3CCR2CYP19A1
SCHEMBL1499268 0.82 HPGD (0.35) GABRA1GABRG2GABRB3CCR2CYP19A1
SCHEMBL3395169 0.82 ALOX5AP (0.36) GABRA1GABRG2GABRB3CCR2NR3C1
SCHEMBL4530176 0.81 ALOX5AP (0.35) GABRA1GABRG2GABRB3CCR2NR3C1
SCHEMBL4538488 0.74 USP2 (0.42) NPSR1
SCHEMBL3395390 0.73 USP2 (0.44) NPSR1
SCHEMBL9804571 0.73 L3MBTL1 (0.39) GABRA1GABRG2GABRB3CYP19A1
SCHEMBL2960873 0.70 CALM1 (0.58) CALM1
SCHEMBL3428803 0.70 NOS3 (0.31) NOS3NOS1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2245123-B1 METHODS FOR PRODUCING ALKYLATED 1,3 BENZENEDIAMINE COMPOUNDS CHEMTURA CORP (US) 2017-07-19 EP disclosed
US-8563489-B2 Alkylated 1,3-benzenediamine compounds and methods for producing same CHEMTURA CORPORATION (US) 2013-10-22 US disclosed
US-20090156449-A1 ALKYLATED 1,3-BENZENEDIAMINE COMPOUNDS AND METHODS FOR PRODUCING SAME LANXESS SOLUTIONS US INC. 2009-06-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090156449-A1 ALKYLATED 1,3-BENZENEDIAMINE COMPOUNDS AND METHODS FOR PRODUCING SAME BBOX1, ABHD5, BRD1 GABRA1 2052/4885GABRG2 1864/4885GABRB3 2196/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.