SCHEMBL4534333

SCHEMBL4534333

COc1cccc(S(=O)(=O)N2CCC(CNC(=O)[C]3CCCCCCC3)C2)c1.[CH2].[CH2]

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 3/20 0.50
ALDH1A1 P00352 6/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
HSD17B10 Q99714 2/20 0.49
HPGD P15428 2/20 0.49
LMNA P02545 1/20 0.49
POLB P06746 1/20 0.49
RAB9A P51151 2/20 0.49
MAPT P10636 2/20 0.47
NPC1 O15118 1/20 0.47
APOBEC3A P31941 1/20 0.47
KMT2A Q03164 1/20 0.47
APOBEC3G Q9HC16 1/20 0.47
GAA P10253 1/20 0.47
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
THRB P10828 1/20 0.46
CHRM5 P08912 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
TP53 P04637 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4543003 0.87 CNR1 (0.48) PKMALDH1A1SMN1; SMN2HSD17B10KMT2A
SCHEMBL4530586 0.87 EPHX2 (0.52) ALDH1A1SMN1; SMN2MAPTKMT2AL3MBTL1
SCHEMBL4539993 0.87 ALDH1A1 (0.51) PKMALDH1A1SMN1; SMN2HSD17B10HPGD
SCHEMBL4535854 0.85 KMT2A (0.47) PKMALDH1A1SMN1; SMN2LMNAMAPT
SCHEMBL4542832 0.85 ALDH1A1 (0.54) PKMALDH1A1SMN1; SMN2HPGDLMNA
SCHEMBL4541789 0.85 NPC1 (0.57) ALDH1A1LMNAPOLBNPC1GAA
SCHEMBL4541160 0.84 CYP19A1 (0.51) ALDH1A1SMN1; SMN2HSD17B10LMNAPOLB
SCHEMBL4537743 0.84 EPHX2 (0.48) ALDH1A1SMN1; SMN2LMNAMAPTKMT2A
SCHEMBL4539847 0.83 USP30 (0.44) POLBMAPTL3MBTL1
SCHEMBL4534329 0.82 PKM (0.49) PKMALDH1A1SMN1; SMN2HSD17B10HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO claimed
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed