SCHEMBL4535503

SCHEMBL4535503

O=C(NCC1CCN(S(=O)(=O)c2ccc(F)cc2)CC1)[C]1CCCCCCC1.[CH2].[CH2]

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.57
KMT2A Q03164 3/20 0.53
EPHX2 P34913 1/20 0.53
POLB P06746 3/20 0.52
KDM4E B2RXH2 2/20 0.52
GAA P10253 1/20 0.52
TP53 P04637 1/20 0.51
L3MBTL1 Q9Y468 2/20 0.50
NAMPT P43490 1/20 0.50
USP5 P45974 1/20 0.50
MEN1 O00255 2/20 0.49
MAPT P10636 1/20 0.49
PKM P14618 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4541337 0.93 CYP3A4 (0.55) ALDH1A1KMT2AEPHX2POLBKDM4E
SCHEMBL4535775 0.89 CYP3A4 (0.61) ALDH1A1KMT2APOLBKDM4EGAA
SCHEMBL4541778 0.89 LMNA (0.58) ALDH1A1KMT2APOLBKDM4EL3MBTL1
SCHEMBL4541041 0.88 ALDH1A1 (0.62) ALDH1A1KMT2AEPHX2KDM4EGAA
SCHEMBL4542840 0.86 PKM (0.57) ALDH1A1KMT2AEPHX2POLBKDM4E
SCHEMBL4534659 0.85 CYP3A4 (0.53) ALDH1A1KMT2AEPHX2POLBKDM4E
SCHEMBL4531162 0.82 KMT2A (0.45) ALDH1A1KMT2AKDM4EL3MBTL1NAMPT
SCHEMBL4535273 0.82 HTT (0.51) ALDH1A1KMT2APOLBKDM4EGAA
SCHEMBL4532819 0.82 ALDH1A1 (0.49) ALDH1A1KMT2AEPHX2POLBKDM4E
SCHEMBL4535343 0.82 HTR7 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed