SCHEMBL4537002

SCHEMBL4537002

COc1cc(S(=O)(=O)N2CCCCC2CNC(=O)C23CC4CC(CC(C4)C2)C3)ccc1O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.44
PAX8 Q06710 1/20 0.43
NCOA1 Q15788 1/20 0.42
NCOA3 Q9Y6Q9 1/20 0.42
ALDH1A1 P00352 1/20 0.41
CA2 P00918 2/20 0.41
DRD2 P14416 2/20 0.41
DRD1 P21728 2/20 0.41
DRD4 P21917 2/20 0.41
DRD3 P35462 2/20 0.41
CA9 Q16790 2/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2D6 P10635 2/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA3 P07451 1/20 0.41
ADRA2A P08913 1/20 0.41
MAPT P10636 1/20 0.41
PTGS1 P23219 1/20 0.41
CA6 P23280 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4540629 0.93 HCRTR1 (0.47) RAB9APAX8ALDH1A1TSHR
SCHEMBL4542350 0.89 RAB9A (0.43) RAB9APAX8NCOA1NCOA3LMNA
SCHEMBL4537060 0.86 ALDH1A1 (0.43) PAX8ALDH1A1DRD2DRD3TSHR
SCHEMBL4539816 0.85 RAB9A (0.60) RAB9APAX8
SCHEMBL4531292 0.85 ALDH1A1 (0.43) RAB9AALDH1A1TSHR
SCHEMBL4537004 0.84 RAB9A (0.49) RAB9APAX8NCOA1NCOA3CA2
SCHEMBL4535257 0.83 RAB9A (0.53) RAB9APAX8NCOA1NCOA3ALDH1A1
SCHEMBL4539052 0.83 ALDH1A1 (0.47) RAB9APAX8ALDH1A1TSHR
SCHEMBL4530967 0.83 HTR7 (0.48) RAB9ADRD2DRD3CYP1A2CYP2D6
SCHEMBL4537168 0.82 RAB9A (0.47) RAB9APAX8LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO claimed
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed