SCHEMBL4537060

SCHEMBL4537060

O=C(NCC1CCCCN1S(=O)(=O)c1ccc(O)c(Cl)c1)C12CC3CC(CC(C3)C1)C2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.43
PSEN1 P49768 2/20 0.41
PSEN2 P49810 2/20 0.41
APH1B Q8WW43 2/20 0.41
NCSTN Q92542 2/20 0.41
APH1A Q96BI3 2/20 0.41
PSENEN Q9NZ42 2/20 0.41
TSHR P16473 2/20 0.40
TP53 P04637 1/20 0.40
HTR7 P34969 2/20 0.39
HTR1A P08908 1/20 0.39
DRD2 P14416 1/20 0.39
HTR1D P28221 1/20 0.39
HTR1B P28222 1/20 0.39
HTR1E P28566 1/20 0.39
ADRA1B P35368 1/20 0.39
DRD3 P35462 1/20 0.39
PAX8 Q06710 1/20 0.39
CASP3 P42574 2/20 0.39
CASP1 P29466 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4542596 0.90 MAPT (0.44) ALDH1A1PSEN1PSEN2APH1BNCSTN
SCHEMBL4535933 0.88 PSEN1 (0.56) ALDH1A1PSEN1PSEN2APH1BNCSTN
SCHEMBL4531292 0.87 ALDH1A1 (0.43) ALDH1A1PSEN1PSEN2APH1BNCSTN
SCHEMBL4541106 0.86 VCAM1 (0.48) ALDH1A1PSEN1PSEN2APH1BNCSTN
SCHEMBL4537002 0.86 RAB9A (0.44) ALDH1A1TSHRDRD2DRD3PAX8
SCHEMBL4538141 0.86 BDKRB1 (0.46) ALDH1A1PSEN1PSEN2APH1BNCSTN
SCHEMBL4541043 0.85 ITGB1 (0.44) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL4534371 0.85 DRD2 (0.41) ALDH1A1PSEN1PSEN2APH1BNCSTN
SCHEMBL4530967 0.85 HTR7 (0.48) HTR7HTR1ADRD2HTR1DHTR1B
SCHEMBL4538787 0.84 PSEN1 (0.51) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO claimed
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed