SCHEMBL4538162

SCHEMBL4538162

COc1ccccc1S(=O)(=O)N1CCCC1CC(=O)NC12CC3CC(CC(C3)C1)C2

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.52
MEN1 O00255 2/20 0.52
CNR2 P34972 4/20 0.47
FAAH O00519 2/20 0.47
LMNA P02545 1/20 0.46
HTT P42858 1/20 0.46
EPHX2 P34913 1/20 0.45
POLB P06746 1/20 0.44
ALDH1A1 P00352 2/20 0.44
HTR1A P08908 1/20 0.42
HTR7 P34969 1/20 0.42
EPHX1 P07099 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4541773 0.87 EPHX2 (0.45) KMT2ACNR2EPHX2ALDH1A1EPHX1
SCHEMBL4536688 0.85 FKBP1A (0.51) KMT2AMEN1CNR2FAAHLMNA
SCHEMBL8067220 0.85 ALDH1A1 (0.54) KMT2APOLBALDH1A1HTR1AHTR7
SCHEMBL4541031 0.85 ALDH1A1 (0.54) KMT2APOLBALDH1A1HTR1AHTR7
SCHEMBL4541290 0.85 HSD11B1 (0.47) KMT2AFAAHLMNAHTTEPHX2
SCHEMBL4537814 0.85 EPHX2 (0.44) KMT2ACNR2EPHX2ALDH1A1EPHX1
SCHEMBL4542819 0.83 RAB9A (0.54) KMT2AEPHX2EPHX1
SCHEMBL4539287 0.83 HCRTR1 (0.48) KMT2AMEN1ALDH1A1EPHX1
SCHEMBL4541277 0.83 HSD11B1 (0.46) KMT2AFAAHLMNAHTTEPHX2
SCHEMBL4542205 0.83 RAB9A (0.52) CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO claimed
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed