Alprenolol

Alprenolol

SCHEMBL4538381

C=CCc1ccccc1OC[C@H](O)CNC(C)C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 9/20 1.00
ADRB1 P08588 9/20 1.00
LMNA P02545 3/20 1.00
HTR1A P08908 2/20 1.00
SLC6A4 P31645 2/20 1.00
ADRA1A P35348 2/20 1.00
CYP1A2 P05177 2/20 1.00
CYP2D6 P10635 2/20 1.00
ADRB3 P13945 2/20 1.00
ADRA2C P18825 1/20 1.00
SLC6A2 P23975 1/20 1.00
BDKRB2 P30411 1/20 1.00
HTR2B P41595 1/20 1.00
KCNH2 Q12809 1/20 1.00
TSHR P16473 1/20 1.00
NFKB1 P19838 1/20 1.00
KDM4E B2RXH2 1/20 0.97
PMP22 Q01453 1/20 0.97
TDP1 Q9NUW8 1/20 0.97
ALDH1A1 P00352 1/20 0.76

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Alprenolol SCHEMBL29414120 1.00 ADRB2 (1.00) ADRB2ADRB1LMNAHTR1ASLC6A4
Alprenolol SCHEMBL34636 1.00 ADRB2 (1.00) ADRB2ADRB1LMNAHTR1ASLC6A4
Alprenolol SCHEMBL29355107 1.00 ADRB2 (1.00) ADRB2ADRB1LMNAHTR1ASLC6A4
Alprenolol SCHEMBL34637 1.00 ADRB2 (1.00) ADRB2ADRB1LMNAHTR1ASLC6A4
Alprenolol SCHEMBL6508231 1.00 ADRB2 (1.00) ADRB2ADRB1LMNAHTR1ASLC6A4
Alprenolol SCHEMBL10762606 0.99 ADRB2 (0.97) ADRB2ADRB1LMNAHTR1ASLC6A4
Alprenolol SCHEMBL29725600 0.99 LMNA (1.00) ADRB2ADRB1LMNAHTR1ASLC6A4
Alprenolol SCHEMBL349102 0.99 LMNA (1.00) ADRB2ADRB1LMNAHTR1ASLC6A4
Alprenolol SCHEMBL349100 0.99 LMNA (1.00) ADRB2ADRB1LMNAHTR1ASLC6A4
Alprenolol SCHEMBL7692100 0.99 ADRB2 (0.97) ADRB2ADRB1LMNAHTR1ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4637708-A2 SEMIFLUORINATED ALKANE COMPOSITIONS COMPRISING HYOSCYAMINE Novaliq GmbH (DE) 2025-10-29 EP claimed
WO-2024133913-A9 SEMIFLUORINATED ALKANE COMPOSITIONS COMPRISING HYOSCYAMINE NOVALIQ GMBH (DE) 2025-03-20 WO claimed
WO-2024133913-A2 SEMIFLUORINATED ALKANE COMPOSITIONS COMPRISING HYOSCYAMINE NOVALIQ GMBH (DE) 2024-06-27 WO claimed
EP-4637708-A2 SEMIFLUORINATED ALKANE COMPOSITIONS COMPRISING HYOSCYAMINE Novaliq GmbH (DE) 2025-10-29 EP disclosed
US-20250179130-A1 METHODS AND SYSTEMS FOR DESIGNING AND/OR CHARACTERIZING SOLUBLE LIPIDATED LIGAND AGENTS ON TARGET THERAPEUTICS LLC 2025-06-05 US disclosed
WO-2024133913-A9 SEMIFLUORINATED ALKANE COMPOSITIONS COMPRISING HYOSCYAMINE NOVALIQ GMBH (DE) 2025-03-20 WO disclosed
US-12060397-B2 Soluble lipidated ligand agents for treating eye inflammation TUFTS MEDICAL CENTER (US) 2024-08-13 US disclosed
WO-2024133913-A2 SEMIFLUORINATED ALKANE COMPOSITIONS COMPRISING HYOSCYAMINE NOVALIQ GMBH (DE) 2024-06-27 WO disclosed
US-20220226310-A1 Bio-Based Medicines and Methods of Increasing Patient Compliance RDE PHARMA 2022-07-21 US disclosed
US-20220135633-A1 METHODS AND SYSTEMS FOR DESIGNING AND/OR CHARACTERIZING SOLUBLE LIPIDATED LIGAND AGENTS ON TARGET THERAPEUTICS LLC 2022-05-05 US disclosed
US-11254720-B2 Methods and systems for designing and/or characterizing soluble lipidated ligand agents ON TARGET THERAPEUTICS LLC (US) 2022-02-22 US disclosed
US-20190135882-A1 Methods and Systems for Designing and/or Characterizing Soluble Lipidated Ligand Agents ON TARGET THERAPEUTICS LLC 2019-05-09 US disclosed
US-10233219-B2 Methods and systems for designing and/or characterizing soluble lipidated ligand agents TUFTS MEDICAL CENTER (US) 2019-03-19 US disclosed
US-20160052982-A1 METHODS AND SYSTEMS FOR DESIGNING AND/OR CHARACTERIZING SOLUBLE LIPIDATED LIGAND AGENTS ON TARGET THERAPEUTICS LLC 2016-02-25 US disclosed
US-20140349969-A1 COMPOUNDS AND METHODS FOR TREATING PAIN AKRON MOLECULES AG (AT) 2014-11-27 US disclosed
EP-2674161-A1 FMO3 inhibitors for treating pain Akron Molecules GmbH (AT) 2013-12-18 EP disclosed
CN-103415286-A Compounds and methods for treating pain AKRON MOLECULES GMBH 2013-11-27 CN disclosed
US-20130252924-A1 Compounds and Methods for Treating Pain AKRON MOLECULES GMBH (AT) 2013-09-26 US disclosed
EP-2637649-A2 COMPOUNDS AND METHODS FOR TREATING PAIN Akron Molecules GmbH (AT) 2013-09-18 EP disclosed
WO-2012062925-A2 COMPOUNDS AND METHODS FOR TREATING PAIN AKRON MOLECULES GMBH (AT) 2012-05-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140349969-A1 COMPOUNDS AND METHODS FOR TREATING PAIN TRPV1, ACHE, OPRL1 ADRB2 237/4885ADRB1 497/4885LMNA 3003/4885
US-20220135633-A1 METHODS AND SYSTEMS FOR DESIGNING AND/OR CHARACTERIZING SOLUBLE LIPIDATED LIGAND AGENTS LDLR, HDLBP, LIPG ADRB2 2941/4885ADRB1 2832/4885LMNA 2571/4885
US-11254720-B2 Methods and systems for designing and/or characterizing soluble lipidated ligand agents LDLR, HDLBP, LIPG ADRB2 2941/4885ADRB1 2832/4885LMNA 2571/4885
US-20220226310-A1 Bio-Based Medicines and Methods of Increasing Patient Compliance PAH, BPGM, TPMT ADRB2 1682/4885ADRB1 1330/4885LMNA 2689/4885
US-20190135882-A1 Methods and Systems for Designing and/or Characterizing Soluble Lipidated Ligand Agents LDLR, HDLBP, LIPG ADRB2 2941/4885ADRB1 2832/4885LMNA 2571/4885
US-20130252924-A1 Compounds and Methods for Treating Pain TRPV1, ACHE, OPRL1 ADRB2 237/4885ADRB1 497/4885LMNA 3003/4885
US-20160052982-A1 METHODS AND SYSTEMS FOR DESIGNING AND/OR CHARACTERIZING SOLUBLE LIPIDATED LIGAND AGENTS LDLR, HDLBP, LIPG ADRB2 2941/4885ADRB1 2832/4885LMNA 2571/4885
US-10233219-B2 Methods and systems for designing and/or characterizing soluble lipidated ligand agents LDLR, HDLBP, LIPG ADRB2 2941/4885ADRB1 2832/4885LMNA 2571/4885
US-20250179130-A1 METHODS AND SYSTEMS FOR DESIGNING AND/OR CHARACTERIZING SOLUBLE LIPIDATED LIGAND AGENTS LDLR, HDLBP, LIPG ADRB2 2941/4885ADRB1 2832/4885LMNA 2571/4885
US-12060397-B2 Soluble lipidated ligand agents for treating eye inflammation LIPG, CD40, LDLR ADRB2 1967/4885ADRB1 1777/4885LMNA 3786/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.